Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 1270
TargetIntermediate conductance calcium-activated potassium channel protein 4(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM314248(US9611232, Example 13)
Affinity DataIC50:  15nMAssay Description:Compounds were tested using a PatchXpress® (Model 7000A, Molecular Devices, Union City Calif.) on CHO cells over-expressing h KCa3.1 at ChanTest Corp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntermediate conductance calcium-activated potassium channel protein 4(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM314285(US9611232, Example 17)
Affinity DataIC50:  15nMAssay Description:Compounds were tested using a PatchXpress® (Model 7000A, Molecular Devices, Union City Calif.) on CHO cells over-expressing h KCa3.1 at ChanTest Corp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntermediate conductance calcium-activated potassium channel protein 4(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM314217(US9611232, Example 11)
Affinity DataIC50:  22nMAssay Description:Compounds were tested using a PatchXpress® (Model 7000A, Molecular Devices, Union City Calif.) on CHO cells over-expressing h KCa3.1 at ChanTest Corp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntermediate conductance calcium-activated potassium channel protein 4(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM314284(US9611232, Example 15)
Affinity DataIC50:  42nMAssay Description:Compounds were tested using a PatchXpress® (Model 7000A, Molecular Devices, Union City Calif.) on CHO cells over-expressing h KCa3.1 at ChanTest Corp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntermediate conductance calcium-activated potassium channel protein 4(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM314215(US9611232, Example 7)
Affinity DataIC50:  45nMAssay Description:Compounds were tested using a PatchXpress® (Model 7000A, Molecular Devices, Union City Calif.) on CHO cells over-expressing h KCa3.1 at ChanTest Corp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntermediate conductance calcium-activated potassium channel protein 4(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM314198((S)-2-(5,5-bis(4-fluorophenyl)-2-oxo-4-phenyloxazo...)
Affinity DataIC50:  58nMAssay Description:Compounds were tested using a PatchXpress® (Model 7000A, Molecular Devices, Union City Calif.) on CHO cells over-expressing h KCa3.1 at ChanTest Corp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntermediate conductance calcium-activated potassium channel protein 4(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM314321(US9611232, Example 32)
Affinity DataIC50:  62nMAssay Description:Compounds were tested using a PatchXpress® (Model 7000A, Molecular Devices, Union City Calif.) on CHO cells over-expressing h KCa3.1 at ChanTest Corp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntermediate conductance calcium-activated potassium channel protein 4(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM314288(US9611232, Example 19)
Affinity DataIC50:  63nMAssay Description:Compounds were tested using a PatchXpress® (Model 7000A, Molecular Devices, Union City Calif.) on CHO cells over-expressing h KCa3.1 at ChanTest Corp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent