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Patent code US9611249

Compile Data Set for Download or QSAR
Found 35 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314399
PNG
(US9611249, Compound 30 | {4-[({[5-(5-methoxypyridi...)
Show SMILES COc1cncc(c1)-c1ccc2[nH]nc(C(=O)NCC3CCN(CC(O)=O)CC3)c2c1
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US Patent
n/an/a 20n/an/an/an/an/an/a



AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM50134187
PNG
(CHEMBL3735506 | US9611249, Compound 8)
Show SMILES COCCN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2cccc(F)c2F)CC1
Show InChI InChI=1S/C23H26F2N4O2/c1-31-12-11-29-9-7-15(8-10-29)14-26-23(30)22-18-13-16(5-6-20(18)27-28-22)17-3-2-4-19(24)21(17)25/h2-6,13,15H,7-12,14H2,1H3,(H,26,30)(H,27,28)
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Similars

US Patent
n/an/a 20n/an/an/an/an/an/a



AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314382
PNG
(N-{[1-(2-methoxyethyl)piperidin-4- yl]methyl}-5-(5...)
Show SMILES COCCN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2cncc(OC)c2)CC1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314398
PNG
(US9611249, Compound 29 | {4-[({[5-(2,3-difluorophe...)
Show SMILES OC(=O)CN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2cccc(F)c2F)CC1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314371
PNG
(N-{[1-(2-methoxyethyl)piperidin-4- yl]methyl}-5-(p...)
Show SMILES COCCN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2cccnc2)CC1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314387
PNG
(N-{[1-(2-methoxyethyl)piperidin-4- yl]methyl}-5-(6...)
Show SMILES COCCN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2ccc(OC)nc2)CC1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314374
PNG
(N-{[1-(2-methoxyethyl)piperidin-4- yl]methyl}-5-(4...)
Show SMILES COCCN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2cnccc2OC)CC1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314378
PNG
(N-{[1-(2-methoxyethyl)piperidin-4- yl]methyl}-5-(6...)
Show SMILES COCCN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2ccc(C)nc2)CC1
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n/an/a 60n/an/an/an/an/an/a



AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314377
PNG
(5-(2-fluorophenyl)-N-{[1-(2- methoxyethyl)piperidi...)
Show SMILES COCCN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2ccccc2F)CC1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314396
PNG
(US9611249, Compound 27 | {4-[({[5-(2,3-dichlorophe...)
Show SMILES OC(=O)CN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2cccc(Cl)c2Cl)CC1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314397
PNG
(US9611249, Compound 28 | {4-[({[5-(3-fluorophenyl)...)
Show SMILES OC(=O)CN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2cccc(F)c2)CC1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314381
PNG
(N-{[1-(2-methoxyethyl)pipendin-4- yl]methyl}-5-phe...)
Show SMILES COCCN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2ccccc2)CC1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314391
PNG
(US9611249, Compound 25 | US9611249, Compound 25b |...)
Show SMILES OC(=O)CN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2cncnc2)CC1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314391
PNG
(US9611249, Compound 25 | US9611249, Compound 25b |...)
Show SMILES OC(=O)CN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2cncnc2)CC1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314384
PNG
(N-{[1-(2-methoxyethyl)piperidin-4- yl]methyl}-5-(4...)
Show SMILES COCCN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2ccc(OC)cc2)CC1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314385
PNG
(N-{[1-(2-methoxyethyl)piperidin-4- yl]methyl}-5-(4...)
Show SMILES COCCN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2ccc(C)cc2)CC1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314388
PNG
(N-{[1-(2-methoxyethyl)piperidin-4- yl]methyl}-5-(2...)
Show SMILES COCCN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2ccccc2C)CC1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314324
PNG
(US9611249, Compound 1 | [4-({[(5-methoxy-1H-indazo...)
Show SMILES COc1ccc2[nH]nc(C(=O)NCC3CCN(CC(O)=O)CC3)c2c1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314370
PNG
(US9611249, Compound 3 | [4-({[(5-methoxy-1H-indazo...)
Show SMILES COc1ccc2[nH]nc(C(=O)NCC3CCN(CCC(O)=O)CC3)c2c1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314407
PNG
(N-[(1-{3-[(2E)-but-2-enoylamino]propyl} piperidin-...)
Show SMILES COc1ccc2[nH]nc(C(=O)NCC3CCN(CCCNC(=O)\C=C\C)CC3)c2c1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314368
PNG
(5-methoxy-N-{[1-(2-methoxyethyl)- piperidin-4-yl]m...)
Show SMILES COCCN1CCC(CNC(=O)c2n[nH]c3ccc(OC)cc23)CC1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314409
PNG
(N-({1-[3-(but-2-ynoylamino)propyl] piperidin-4-yl}...)
Show SMILES COc1ccc2[nH]nc(C(=O)NCC3CCN(CCCNC(=O)C#CC)CC3)c2c1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314383
PNG
(5-(4-hydroxyphenyl)-N-{[1-(2- methoxyethyl)piperid...)
Show SMILES COCCN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2ccc(O)cc2)CC1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314395
PNG
(US9611249, Compound 26 | {4-[({[5-(3,5-Dimethyliso...)
Show SMILES Cc1noc(C)c1-c1ccc2[nH]nc(C(=O)NCC3CCN(CC(O)=O)CC3)c2c1
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AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314408
PNG
(5-methoxy-N-({1-[3-(propanoylamino) propyl]piperid...)
Show SMILES CCC(=O)NCCCN1CCC(CNC(=O)c2n[nH]c3ccc(OC)cc23)CC1
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n/an/a 950n/an/an/an/an/an/a



AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314400
PNG
(US9611249, Compound 31 | [4-({[(5-ethyl-1H-indazol...)
Show SMILES CCc1ccc2[nH]nc(C(=O)NCC3CCN(CC(O)=O)CC3)c2c1
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n/an/a 960n/an/an/an/an/an/a



AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314406
PNG
(N-({1-[3-(butanoylamino)propyl] piperidin-4-yl}met...)
Show SMILES CCCC(=O)NCCCN1CCC(CNC(=O)c2n[nH]c3ccc(OC)cc23)CC1
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n/an/a 970n/an/an/an/an/an/a



AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314390
PNG
(4-[4-({[(5-methoxy-1H-indazol-3-yl) carbonyl]amino...)
Show SMILES COc1ccc2[nH]nc(C(=O)NCC3CCN(CCCC(O)=O)CC3)c2c1
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n/an/a 1.03E+3n/an/an/an/an/an/a



AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314402
PNG
(US9611249, Compound 33 | {4-[({[5-(3,6-dihydro-2H-...)
Show SMILES OC(=O)CN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)C2=CCOCC2)CC1
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n/an/a 1.04E+3n/an/an/an/an/an/a



AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314389
PNG
(5-(2-ethoxy-4,5-difluorophenyl)-N- {[1-(2-methoxye...)
Show SMILES CCOc1cc(F)c(F)cc1-c1ccc2[nH]nc(C(=O)NCC3CCN(CCOC)CC3)c2c1
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n/an/a 1.06E+3n/an/an/an/an/an/a



AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314403
PNG
(US9611249, Compound 34 | [4-({[(5-cyclohexyl-1H-in...)
Show SMILES OC(=O)CN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)C2CCCCC2)CC1
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n/an/a 1.07E+3n/an/an/an/an/an/a



AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314386
PNG
(N-{[1-(2-methoxyethyl)piperidin-4- yl]methyl}-5-(2...)
Show SMILES COCCN1CCC(CNC(=O)c2n[nH]c3ccc(cc23)-c2cccnc2OC)CC1
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n/an/a 1.40E+3n/an/an/an/an/an/a



AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314404
PNG
(US9611249, Compound 35 | [4-({[(5-pentyl-1H-indazo...)
Show SMILES CCCCCc1ccc2[nH]nc(C(=O)NCC3CCN(CC(O)=O)CC3)c2c1
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n/an/a 2.04E+3n/an/an/an/an/an/a



AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314405
PNG
(5-methoxy-N-[(1-{3- [(phenylcarbonyl)amino]propyl}...)
Show SMILES COc1ccc2[nH]nc(C(=O)NCC3CCN(CCCNC(=O)c4ccccc4)CC3)c2c1
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n/an/a 3.42E+3n/an/an/an/an/an/a



AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
Glycogen synthase kinase-3 beta


(Homo sapiens (human))
BDBM314401
PNG
(US9611249, Compound 32 | {4-[({[5-(propan-2-yl)-1H...)
Show SMILES CC(C)c1ccc2[nH]nc(C(=O)NCC3CCN(CC(O)=O)CC3)c2c1
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n/an/a 3.91E+3n/an/an/an/an/an/a



AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A.

US Patent


Assay Description
Activity on human GSK-3β was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screen...


US Patent US9611249 (2017)

More data for this
Ligand-Target Pair
* indicates data uncertainty>20%