Compile Data Set for Download or QSAR
maximum 50k data
Found 67 Enz. Inhib. hit(s) with all data for entry = 1333
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317482(4-(4-((1s,4s)-4-hydroxy-4- methylcyclohexyloxy)-5-...)
Affinity DataIC50:  1.15nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317480(4-(4-isopropoxy-5-(4- (methylcarbamoyl)phenyl)-7H-...)
Affinity DataIC50:  1.42nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317482(4-(4-((1s,4s)-4-hydroxy-4- methylcyclohexyloxy)-5-...)
Affinity DataIC50:  1.43nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317475(3-cyano-N-methyl-4-(5-(2- methylbenzo[d]oxazol-6-y...)
Affinity DataIC50:  1.47nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317466(4-(4-methoxy-5-(pyridin-4-yl)- 7H-pyrrolo[2,3-d]py...)
Affinity DataIC50: <1.5nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317467(3-methoxy-N-methyl-4-(5-(2- methylbenzo[d]oxazol-6...)
Affinity DataIC50:  1.68nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317471((S)-3-chloro-N-methyl-4-(5-(2- methylbenzo[d]oxazo...)
Affinity DataIC50:  1.68nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317485(3-chloro-N-methyl-4-(5-(1- methyl-1H-pyrazol-4-yl)...)
Affinity DataIC50:  1.90nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317465(4-(4-(cyclopentyloxy)-5-(4- (methylcarbamoyl)pheny...)
Affinity DataIC50:  1.91nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317483(3-chloro-N-methyl-4-(5-(4- (methylcarbamoyl)phenyl...)
Affinity DataIC50:  2.10nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317473(4-(5-(4-(1H-imidazol-2- yl)phenyl)-4-(tetrahydro-2...)
Affinity DataIC50:  2.12nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317468(4-(4-(cyclopentyloxy)-5-(2- methylbenzo[d]oxazol-6...)
Affinity DataIC50:  2.13nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317471((S)-3-chloro-N-methyl-4-(5-(2- methylbenzo[d]oxazo...)
Affinity DataIC50:  2.27nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317469(3-methoxy-4-(4-methoxy-5-(6- methoxypyridin-3-yl)-...)
Affinity DataIC50:  2.29nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317475(3-cyano-N-methyl-4-(5-(2- methylbenzo[d]oxazol-6-y...)
Affinity DataIC50:  2.32nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317479(4-(4-cyclobutoxy-5-(4- (methylcarbamoyl)phenyl)-7H...)
Affinity DataIC50:  2.35nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317465(4-(4-(cyclopentyloxy)-5-(4- (methylcarbamoyl)pheny...)
Affinity DataIC50:  2.38nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317472(N,3-dimethyl-4-(5-(2- methylbenzo[d]oxazol-6-yl)-4...)
Affinity DataIC50:  2.45nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317474(4-(4-cyclopropoxy-5-(2- methylbenzo[d]oxazol-6-yl)...)
Affinity DataIC50:  2.96nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317485(3-chloro-N-methyl-4-(5-(1- methyl-1H-pyrazol-4-yl)...)
Affinity DataIC50:  3.29nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317468(4-(4-(cyclopentyloxy)-5-(2- methylbenzo[d]oxazol-6...)
Affinity DataIC50:  3.38nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317467(3-methoxy-N-methyl-4-(5-(2- methylbenzo[d]oxazol-6...)
Affinity DataIC50:  3.5nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317476(N-methyl-4-(5-(2- methylbenzo[d]oxazol-6-yl)-4- (t...)
Affinity DataIC50:  3.65nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317470(3-chloro-N-methyl-4-(5-(2- methylbenzo[d]oxazol-6-...)
Affinity DataIC50:  4.12nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317460(4-(5-(4-hydroxyphenyl)-4- (tetrahydro-2H-pyran-4-y...)
Affinity DataIC50:  4.33nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317478(4-(4-(cyclopentyloxy)-5-(2- methylbenzo[d]oxazol-6...)
Affinity DataIC50:  4.54nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317466(4-(4-methoxy-5-(pyridin-4-yl)- 7H-pyrrolo[2,3-d]py...)
Affinity DataIC50:  4.56nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317469(3-methoxy-4-(4-methoxy-5-(6- methoxypyridin-3-yl)-...)
Affinity DataIC50:  5.14nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317481(4-(4-cyclobutoxy-5-(2- methylbenzo[d]oxazol-6-yl)-...)
Affinity DataIC50:  5.92nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317481(4-(4-cyclobutoxy-5-(2- methylbenzo[d]oxazol-6-yl)-...)
Affinity DataIC50:  7nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317477(4-(4-(cyclopentyloxy)-5-(2- methylbenzo[d]oxazol-6...)
Affinity DataIC50:  8.06nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317462(4-(4-(cyclopentyloxy)-5-(2- methylbenzo[d]oxazol-6...)
Affinity DataIC50:  8.17nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317476(N-methyl-4-(5-(2- methylbenzo[d]oxazol-6-yl)-4- (t...)
Affinity DataIC50:  9.41nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317477(4-(4-(cyclopentyloxy)-5-(2- methylbenzo[d]oxazol-6...)
Affinity DataIC50:  10.4nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317484(3-chloro-4-(4-(cyclopentyloxy)-5- (2-methylbenzo[d...)
Affinity DataIC50:  11.6nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317484(3-chloro-4-(4-(cyclopentyloxy)-5- (2-methylbenzo[d...)
Affinity DataIC50:  12.5nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317463(4-(4-(cyclopentyloxy)-5-(6- methoxypyridin-3-yl)-7...)
Affinity DataIC50:  13.3nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317462(4-(4-(cyclopentyloxy)-5-(2- methylbenzo[d]oxazol-6...)
Affinity DataIC50:  14nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317464(4-(4-(cyclopentyloxy)-5-(6- ethoxypyridin-3-yl)-7H...)
Affinity DataIC50:  16nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317458(4-(4-(cyclopentylamino)-5-(4- hydroxyphenyl)-7H-py...)
Affinity DataIC50:  26nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317470(3-chloro-N-methyl-4-(5-(2- methylbenzo[d]oxazol-6-...)
Affinity DataIC50:  29.1nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317465(4-(4-(cyclopentyloxy)-5-(4- (methylcarbamoyl)pheny...)
Affinity DataIC50:  34nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317456(4-(4-(cyclopentyloxy)-5-(4- hydroxyphenyl)-7H-pyrr...)
Affinity DataIC50:  34.9nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317472(N,3-dimethyl-4-(5-(2- methylbenzo[d]oxazol-6-yl)-4...)
Affinity DataIC50:  40.1nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317466(4-(4-methoxy-5-(pyridin-4-yl)- 7H-pyrrolo[2,3-d]py...)
Affinity DataIC50:  41.5nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317455(4-(4-(cyclopentyloxy)-5-(4- hydroxyphenyl)-7H-pyrr...)
Affinity DataIC50:  53.9nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317465(4-(4-(cyclopentyloxy)-5-(4- (methylcarbamoyl)pheny...)
Affinity DataIC50:  58.6nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317482(4-(4-((1s,4s)-4-hydroxy-4- methylcyclohexyloxy)-5-...)
Affinity DataIC50:  59.3nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317460(4-(5-(4-hydroxyphenyl)-4- (tetrahydro-2H-pyran-4-y...)
Affinity DataIC50:  82.4nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Signal Pharmaceuticals

US Patent
LigandPNGBDBM317475(3-cyano-N-methyl-4-(5-(2- methylbenzo[d]oxazol-6-y...)
Affinity DataIC50:  82.8nMAssay Description:The kinase activity is measured using a radioactivity based kinase assay, which measures the incorporation of a radioactively labeled phosphate moiet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 67 total ) | Next | Last >>
Jump to: