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Patent code US9663460

Compile Data Set for Download or QSAR

Found 209 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327373
PNG
(N-(5-chloro-2-{[(2-fluoropyridin-3-yl)methyl]-sulf...)
Show SMILES Fc1ncccc1CS(=O)c1ccc(Cl)cc1NS(=O)(=O)c1cc2ccccc2o1
Show InChI InChI=1S/C20H14ClFN2O4S2/c21-15-7-8-18(29(25)12-14-5-3-9-23-20(14)22)16(11-15)24-30(26,27)19-10-13-4-1-2-6-17(13)28-19/h1-11,24H,12H2
PDB

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UniProtKB/SwissProt

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UniChem
US Patent
n/an/a 79n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327290
PNG
(N-[2-({2-[(aminocarbonyl)amino]ethyl}thio)-5-chlor...)
Show SMILES NC(=O)NCCSc1ccc(Cl)cc1NS(=O)(=O)c1cc2ccccc2o1
Show InChI InChI=1S/C17H16ClN3O4S2/c18-12-5-6-15(26-8-7-20-17(19)22)13(10-12)21-27(23,24)16-9-11-3-1-2-4-14(11)25-16/h1-6,9-10,21H,7-8H2,(H3,19,20,22)
PDB

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UniProtKB/SwissProt

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UniChem
US Patent
n/an/a 80n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327343
PNG
(N-(2-{[(2-aminopyridin-4-yl)methyl]thio}-5-chlorop...)
Show SMILES Nc1cc(CSc2ccc(Cl)cc2NS(=O)(=O)c2cc3ccccc3o2)ccn1
Show InChI InChI=1S/C20H16ClN3O3S2/c21-15-5-6-18(28-12-13-7-8-23-19(22)9-13)16(11-15)24-29(25,26)20-10-14-3-1-2-4-17(14)27-20/h1-11,24H,12H2,(H2,22,23)
PDB

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US Patent
n/an/a 80n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327286
PNG
(N-{5-chloro-2-[(1H-imidazol-4-ylmethyl)-sulfonyl]p...)
Show SMILES Clc1ccc(c(NS(=O)(=O)c2cc3ccccc3o2)c1)S(=O)(=O)Cc1c[nH]cn1
Show InChI InChI=1S/C18H14ClN3O5S2/c19-13-5-6-17(28(23,24)10-14-9-20-11-21-14)15(8-13)22-29(25,26)18-7-12-3-1-2-4-16(12)27-18/h1-9,11,22H,10H2,(H,20,21)
PDB

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US Patent
n/an/a 81n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327323
PNG
(N-(2-{[(2-amino-1,3-thiazol-4-yl)methyl]sulfonyl}-...)
Show SMILES Nc1nc(CS(=O)(=O)c2ccc(Cl)cc2NS(=O)(=O)c2cc3ccccc3o2)cs1
Show InChI InChI=1S/C18H14ClN3O5S3/c19-12-5-6-16(29(23,24)10-13-9-28-18(20)21-13)14(8-12)22-30(25,26)17-7-11-3-1-2-4-15(11)27-17/h1-9,22H,10H2,(H2,20,21)
PDB

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US Patent
n/an/a 83n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327392
PNG
(N-{2-[(3-aminobenzyl)sulfinyl]-5-methoxy-phenyl}-1...)
Show SMILES COc1ccc(c(NS(=O)(=O)c2cc3ccccc3o2)c1)S(=O)Cc1cccc(N)c1
Show InChI InChI=1S/C22H20N2O5S2/c1-28-18-9-10-21(30(25)14-15-5-4-7-17(23)11-15)19(13-18)24-31(26,27)22-12-16-6-2-3-8-20(16)29-22/h2-13,24H,14,23H2,1H3
PDB

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n/an/a 85n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327273
PNG
(4-chloro-N-[5-chloro-2-(methylsulfinyl)phenyl]-2-f...)
Show SMILES CS(=O)c1ccc(Cl)cc1NS(=O)(=O)c1ccc(Cl)cc1F
Show InChI InChI=1S/C13H10Cl2FNO3S2/c1-21(18)12-4-2-9(15)7-11(12)17-22(19,20)13-5-3-8(14)6-10(13)16/h2-7,17H,1H3
PDB

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US Patent
n/an/a 85n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327239
PNG
(4-chloro-N-[5-chloro-2-(ethylsulfonyl)phenyl]-3-(t...)
Show SMILES CCS(=O)(=O)c1ccc(Cl)cc1NS(=O)(=O)c1ccc(Cl)c(c1)C(F)(F)F
Show InChI InChI=1S/C15H12Cl2F3NO4S2/c1-2-26(22,23)14-6-3-9(16)7-13(14)21-27(24,25)10-4-5-12(17)11(8-10)15(18,19)20/h3-8,21H,2H2,1H3
PDB

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US Patent
n/an/a 88n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327398
PNG
(N-{2-[(4-aminobenzyl)sulfonyl]-5-chlorophenyl}-1-b...)
Show SMILES Nc1ccc(CS(=O)(=O)c2ccc(Cl)cc2NS(=O)(=O)c2cc3ccccc3o2)cc1
Show InChI InChI=1S/C21H17ClN2O5S2/c22-16-7-10-20(30(25,26)13-14-5-8-17(23)9-6-14)18(12-16)24-31(27,28)21-11-15-3-1-2-4-19(15)29-21/h1-12,24H,13,23H2
PDB

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n/an/a 90n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327224
PNG
(4-chloro-N-{5-chloro-2-[(pyridin-2-ylmethyl)sulfin...)
Show SMILES FC(F)(F)c1cc(ccc1Cl)S(=O)(=O)Nc1cc(Cl)ccc1S(=O)Cc1ccccn1
Show InChI InChI=1S/C19H13Cl2F3N2O3S2/c20-12-4-7-18(30(27)11-13-3-1-2-8-25-13)17(9-12)26-31(28,29)14-5-6-16(21)15(10-14)19(22,23)24/h1-10,26H,11H2
PDB

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n/an/a 92n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327223
PNG
(4-chloro-N-{5-chloro-2-[(pyridin-3-ylmethyl)thio]-...)
Show SMILES FC(F)(F)c1cc(ccc1Cl)S(=O)(=O)Nc1cc(Cl)ccc1SCc1cccnc1
Show InChI InChI=1S/C19H13Cl2F3N2O2S2/c20-13-3-6-18(29-11-12-2-1-7-25-10-12)17(8-13)26-30(27,28)14-4-5-16(21)15(9-14)19(22,23)24/h1-10,26H,11H2
PDB

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UniChem
US Patent
n/an/a 94n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327372
PNG
(N-(5-chloro-2-{[(2-fluoropyridin-3-yl)methyl]-thio...)
Show SMILES Fc1ncccc1CSc1ccc(Cl)cc1NS(=O)(=O)c1cc2ccccc2o1
Show InChI InChI=1S/C20H14ClFN2O3S2/c21-15-7-8-18(28-12-14-5-3-9-23-20(14)22)16(11-15)24-29(25,26)19-10-13-4-1-2-6-17(13)27-19/h1-11,24H,12H2
PDB

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n/an/a 94n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327220
PNG
(4-chloro-N-{5-chloro-2-[(2-hydroxyethyl)sulfonyl]-...)
Show SMILES OCCS(=O)(=O)c1ccc(Cl)cc1NS(=O)(=O)c1ccc(Cl)c(c1)C(F)(F)F
Show InChI InChI=1S/C15H12Cl2F3NO5S2/c16-9-1-4-14(27(23,24)6-5-22)13(7-9)21-28(25,26)10-2-3-12(17)11(8-10)15(18,19)20/h1-4,7-8,21-22H,5-6H2
PDB

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n/an/a 95n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327230
PNG
(3-{[4-chloro-2-({[4-chloro-3-(trifluoromethyl)-phe...)
Show SMILES CN(C)C(=O)CCS(=O)c1ccc(Cl)cc1NS(=O)(=O)c1ccc(Cl)c(c1)C(F)(F)F
Show InChI InChI=1S/C18H17Cl2F3N2O4S2/c1-25(2)17(26)7-8-30(27)16-6-3-11(19)9-15(16)24-31(28,29)12-4-5-14(20)13(10-12)18(21,22)23/h3-6,9-10,24H,7-8H2,1-2H3
PDB

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n/an/a 96n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327396
PNG
(N-{2-[(2-aminobenzyl)thio]-5-chlorophenyl}-1-benzo...)
Show SMILES Nc1ccccc1CSc1ccc(Cl)cc1NS(=O)(=O)c1cc2ccccc2o1
Show InChI InChI=1S/C21H17ClN2O3S2/c22-16-9-10-20(28-13-15-6-1-3-7-17(15)23)18(12-16)24-29(25,26)21-11-14-5-2-4-8-19(14)27-21/h1-12,24H,13,23H2
PDB

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n/an/a 100n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327235
PNG
(4-chloro-N-{5-chloro-2-[(3-hydroxycyclopentyl)sulf...)
Show SMILES OC1CCC(C1)S(=O)c1ccc(Cl)cc1NS(=O)(=O)c1ccc(Cl)c(c1)C(F)(F)F
Show InChI InChI=1S/C18H16Cl2F3NO4S2/c19-10-1-6-17(29(26)12-3-2-11(25)8-12)16(7-10)24-30(27,28)13-4-5-15(20)14(9-13)18(21,22)23/h1,4-7,9,11-12,24-25H,2-3,8H2
PDB

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n/an/a 107n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327221
PNG
(US9663460, Example 8 | methyl 3-{[4-chloro-2-({[4-...)
Show SMILES COC(=O)CCS(=O)c1ccc(Cl)cc1NS(=O)(=O)c1ccc(Cl)c(c1)C(F)(F)F
Show InChI InChI=1S/C17H14Cl2F3NO5S2/c1-28-16(24)6-7-29(25)15-5-2-10(18)8-14(15)23-30(26,27)11-3-4-13(19)12(9-11)17(20,21)22/h2-5,8-9,23H,6-7H2,1H3
PDB

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n/an/a 108n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327353
PNG
(N-{5-chloro-2-[(3-hydroxybenzyl)sulfinyl]phenyl}-1...)
Show SMILES Oc1cccc(CS(=O)c2ccc(Cl)cc2NS(=O)(=O)c2cc3ccccc3o2)c1
Show InChI InChI=1S/C21H16ClNO5S2/c22-16-8-9-20(29(25)13-14-4-3-6-17(24)10-14)18(12-16)23-30(26,27)21-11-15-5-1-2-7-19(15)28-21/h1-12,23-24H,13H2
PDB

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n/an/a 112n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327225
PNG
(4-chloro-N-{5-chloro-2-[(pyridin-3-ylmethyl)sulfin...)
Show SMILES FC(F)(F)c1cc(ccc1Cl)S(=O)(=O)Nc1cc(Cl)ccc1S(=O)Cc1cccnc1
Show InChI InChI=1S/C19H13Cl2F3N2O3S2/c20-13-3-6-18(30(27)11-12-2-1-7-25-10-12)17(8-13)26-31(28,29)14-4-5-16(21)15(9-14)19(22,23)24/h1-10,26H,11H2
PDB

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n/an/a 112n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327407
PNG
(N-{2-[(3-aminobenzyl)sulfinyl]-5-chlorophenyl}-4-c...)
Show SMILES Nc1cccc(CS(=O)c2ccc(Cl)cc2NS(=O)(=O)c2ccc(Cl)cc2F)c1
Show InChI InChI=1S/C19H15Cl2FN2O3S2/c20-13-5-7-19(16(22)9-13)29(26,27)24-17-10-14(21)4-6-18(17)28(25)11-12-2-1-3-15(23)8-12/h1-10,24H,11,23H2
PDB

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n/an/a 113n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327400
PNG
(N-{2-[(2-aminobenzyl)sulfinyl]-5-chlorophenyl}-1-b...)
Show SMILES Nc1ccccc1CS(=O)c1ccc(Cl)cc1NS(=O)(=O)c1cc2ccccc2o1
Show InChI InChI=1S/C21H17ClN2O4S2/c22-16-9-10-20(29(25)13-15-6-1-3-7-17(15)23)18(12-16)24-30(26,27)21-11-14-5-2-4-8-19(14)28-21/h1-12,24H,13,23H2
PDB

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n/an/a 115n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327315
PNG
(4-bromo-N-[5-chloro-2-(methylsulfinyl)phenyl]benze...)
Show SMILES CS(=O)c1ccc(Cl)cc1NS(=O)(=O)c1ccc(Br)cc1
Show InChI InChI=1S/C13H11BrClNO3S2/c1-20(17)13-7-4-10(15)8-12(13)16-21(18,19)11-5-2-9(14)3-6-11/h2-8,16H,1H3
PDB

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US Patent
n/an/a 116n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327270
PNG
(3-chloro-N-[5-chloro-2-(methylsulfonyl)phenyl]-2-f...)
Show SMILES CS(=O)(=O)c1ccc(Cl)cc1NS(=O)(=O)c1cccc(Cl)c1F
Show InChI InChI=1S/C13H10Cl2FNO4S2/c1-22(18,19)11-6-5-8(14)7-10(11)17-23(20,21)12-4-2-3-9(15)13(12)16/h2-7,17H,1H3
PDB

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n/an/a 116n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327251
PNG
(2-{[4-chloro-2-({[4-chloro-3-(trifluoromethyl)-phe...)
Show SMILES CN(C)C(=O)CSc1ccc(Cl)cc1NS(=O)(=O)c1ccc(Cl)c(c1)C(F)(F)F
Show InChI InChI=1S/C17H15Cl2F3N2O3S2/c1-24(2)16(25)9-28-15-6-3-10(18)7-14(15)23-29(26,27)11-4-5-13(19)12(8-11)17(20,21)22/h3-8,23H,9H2,1-2H3
PDB

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n/an/a 118n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327378
PNG
(N-[2-(benzylthio)-5-chlorophenyl]-1-benzofuran-2-s...)
Show SMILES Clc1ccc(SCc2ccccc2)c(NS(=O)(=O)c2cc3ccccc3o2)c1
Show InChI InChI=1S/C21H16ClNO3S2/c22-17-10-11-20(27-14-15-6-2-1-3-7-15)18(13-17)23-28(24,25)21-12-16-8-4-5-9-19(16)26-21/h1-13,23H,14H2
PDB

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n/an/a 129n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327401
PNG
(N-{2-[(2-aminobenzyl)sulfonyl]-5-chlorophenyl}-1-b...)
Show SMILES Nc1ccccc1CS(=O)(=O)c1ccc(Cl)cc1NS(=O)(=O)c1cc2ccccc2o1
Show InChI InChI=1S/C21H17ClN2O5S2/c22-16-9-10-20(30(25,26)13-15-6-1-3-7-17(15)23)18(12-16)24-31(27,28)21-11-14-5-2-4-8-19(14)29-21/h1-12,24H,13,23H2
PDB

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n/an/a 129n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327216
PNG
(4-chloro-N-[5-chloro-2-(methylthio)phenyl]-3-(trif...)
Show SMILES CSc1ccc(Cl)cc1NS(=O)(=O)c1ccc(Cl)c(c1)C(F)(F)F
Show InChI InChI=1S/C14H10Cl2F3NO2S2/c1-23-13-5-2-8(15)6-12(13)20-24(21,22)9-3-4-11(16)10(7-9)14(17,18)19/h2-7,20H,1H3
PDB

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n/an/a 134n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327226
PNG
(US9663460, Example 13 | ethyl {[4-chloro-2-({[4-ch...)
Show SMILES CCOC(=O)CS(=O)c1ccc(Cl)cc1NS(=O)(=O)c1ccc(Cl)c(c1)C(F)(F)F
Show InChI InChI=1S/C17H14Cl2F3NO5S2/c1-2-28-16(24)9-29(25)15-6-3-10(18)7-14(15)23-30(26,27)11-4-5-13(19)12(8-11)17(20,21)22/h3-8,23H,2,9H2,1H3
PDB

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n/an/a 141n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327219
PNG
(4-chloro-N-{5-chloro-2-[(2-hydroxyethyl)sulfinyl]-...)
Show SMILES OCCS(=O)c1ccc(Cl)cc1NS(=O)(=O)c1ccc(Cl)c(c1)C(F)(F)F
Show InChI InChI=1S/C15H12Cl2F3NO4S2/c16-9-1-4-14(26(23)6-5-22)13(7-9)21-27(24,25)10-2-3-12(17)11(8-10)15(18,19)20/h1-4,7-8,21-22H,5-6H2
PDB

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n/an/a 146n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327287
PNG
(3-({2-[(1-benzofuran-2-ylsulfonyl)amino]-4-chlorop...)
Show SMILES CN(C)C(=O)CCSc1ccc(Cl)cc1NS(=O)(=O)c1cc2ccccc2o1
Show InChI InChI=1S/C19H19ClN2O4S2/c1-22(2)18(23)9-10-27-17-8-7-14(20)12-15(17)21-28(24,25)19-11-13-5-3-4-6-16(13)26-19/h3-8,11-12,21H,9-10H2,1-2H3
PDB

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n/an/a 146n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327395
PNG
(N-{5-chloro-2-[(4-nitrobenzyl)thio]phenyl}-1-benzo...)
Show SMILES [O-][N+](=O)c1ccc(CSc2ccc(Cl)cc2NS(=O)(=O)c2cc3ccccc3o2)cc1
Show InChI InChI=1S/C21H15ClN2O5S2/c22-16-7-10-20(30-13-14-5-8-17(9-6-14)24(25)26)18(12-16)23-31(27,28)21-11-15-3-1-2-4-19(15)29-21/h1-12,23H,13H2
PDB

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ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327410
PNG
(N-{5-chloro-2-[(pyrimidin-2-ylmethyl)sulfonyl]-phe...)
Show SMILES Clc1ccc(c(NS(=O)(=O)c2cc3ccccc3o2)c1)S(=O)(=O)Cc1ncccn1
Show InChI InChI=1S/C19H14ClN3O5S2/c20-14-6-7-17(29(24,25)12-18-21-8-3-9-22-18)15(11-14)23-30(26,27)19-10-13-4-1-2-5-16(13)28-19/h1-11,23H,12H2
PDB

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ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327365
PNG
(N-{5-chloro-2-[(2-pyridin-2-ylethyl)sulfinyl]-phen...)
Show SMILES Clc1ccc(c(NS(=O)(=O)c2cc3ccccc3o2)c1)S(=O)CCc1ccccn1
Show InChI InChI=1S/C21H17ClN2O4S2/c22-16-8-9-20(29(25)12-10-17-6-3-4-11-23-17)18(14-16)24-30(26,27)21-13-15-5-1-2-7-19(15)28-21/h1-9,11,13-14,24H,10,12H2
PDB

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ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327218
PNG
(4-chloro-N-{5-chloro-2-[(2-hydroxyethyl)thio]-phen...)
Show SMILES OCCSc1ccc(Cl)cc1NS(=O)(=O)c1ccc(Cl)c(c1)C(F)(F)F
Show InChI InChI=1S/C15H12Cl2F3NO3S2/c16-9-1-4-14(25-6-5-22)13(7-9)21-26(23,24)10-2-3-12(17)11(8-10)15(18,19)20/h1-4,7-8,21-22H,5-6H2
PDB

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ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327249
PNG
(4-chloro-N-[5-chloro-2-(methylsulfonyl)phenyl]benz...)
Show SMILES CS(=O)(=O)c1ccc(Cl)cc1NS(=O)(=O)c1ccc(Cl)cc1
Show InChI InChI=1S/C13H11Cl2NO4S2/c1-21(17,18)13-7-4-10(15)8-12(13)16-22(19,20)11-5-2-9(14)3-6-11/h2-8,16H,1H3
PDB

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ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327279
PNG
(4-chloro-N-{5-chloro-2-[(1H-imidazol-4-ylmethyl)su...)
Show SMILES FC(F)(F)c1cc(ccc1Cl)S(=O)(=O)Nc1cc(Cl)ccc1S(=O)Cc1c[nH]cn1
Show InChI InChI=1S/C17H12Cl2F3N3O3S2/c18-10-1-4-16(29(26)8-11-7-23-9-24-11)15(5-10)25-30(27,28)12-2-3-14(19)13(6-12)17(20,21)22/h1-7,9,25H,8H2,(H,23,24)
PDB

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ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327419
PNG
(N-{2-[(3-aminobenzyl)sulfinyl]-5-chlorophenyl}-3-c...)
Show SMILES Nc1cccc(CS(=O)c2ccc(Cl)cc2NS(=O)(=O)c2cccc(Cl)c2)c1
Show InChI InChI=1S/C19H16Cl2N2O3S2/c20-14-4-2-6-17(10-14)28(25,26)23-18-11-15(21)7-8-19(18)27(24)12-13-3-1-5-16(22)9-13/h1-11,23H,12,22H2
PDB

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ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327417
PNG
(N-{2-[(3-aminobenzyl)sulfinyl]-5-chlorophenyl}-4-c...)
Show SMILES Nc1cccc(CS(=O)c2ccc(Cl)cc2NS(=O)(=O)c2ccc(Cl)cc2)c1
Show InChI InChI=1S/C19H16Cl2N2O3S2/c20-14-4-7-17(8-5-14)28(25,26)23-18-11-15(21)6-9-19(18)27(24)12-13-2-1-3-16(22)10-13/h1-11,23H,12,22H2
PDB

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ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327288
PNG
(3-({2-[(1-benzofuran-2-ylsulfonyl)amino]-4-chlorop...)
Show SMILES CN(C)C(=O)CCS(=O)c1ccc(Cl)cc1NS(=O)(=O)c1cc2ccccc2o1
Show InChI InChI=1S/C19H19ClN2O5S2/c1-22(2)18(23)9-10-28(24)17-8-7-14(20)12-15(17)21-29(25,26)19-11-13-5-3-4-6-16(13)27-19/h3-8,11-12,21H,9-10H2,1-2H3
PDB

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ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327276
PNG
(4-chloro-N-{5-chloro-2-[(1H-imidazol-2-ylmethyl)su...)
Show SMILES FC(F)(F)c1cc(ccc1Cl)S(=O)(=O)Nc1cc(Cl)ccc1S(=O)Cc1ncc[nH]1
Show InChI InChI=1S/C17H12Cl2F3N3O3S2/c18-10-1-4-15(29(26)9-16-23-5-6-24-16)14(7-10)25-30(27,28)11-2-3-13(19)12(8-11)17(20,21)22/h1-8,25H,9H2,(H,23,24)
PDB

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ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327272
PNG
(4-chloro-N-[5-chloro-2-(methylsulfonyl)phenyl]-2-f...)
Show SMILES CS(=O)(=O)c1ccc(Cl)cc1NS(=O)(=O)c1ccc(Cl)cc1F
Show InChI InChI=1S/C13H10Cl2FNO4S2/c1-22(18,19)13-5-3-9(15)7-11(13)17-23(20,21)12-4-2-8(14)6-10(12)16/h2-7,17H,1H3
PDB

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ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327387
PNG
(N-{2-[(3-aminobenzyl)sulfonyl]-5-methoxyphenyl}-1-...)
Show SMILES COc1ccc(c(NS(=O)(=O)c2cc3ccccc3o2)c1)S(=O)(=O)Cc1cccc(N)c1
Show InChI InChI=1S/C22H20N2O6S2/c1-29-18-9-10-21(31(25,26)14-15-5-4-7-17(23)11-15)19(13-18)24-32(27,28)22-12-16-6-2-3-8-20(16)30-22/h2-13,24H,14,23H2,1H3
PDB

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ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327246
PNG
(N-[5-chloro-2-(methylsulfinyl)phenyl]-4-methyl-3-n...)
Show SMILES Cc1ccc(cc1[N+]([O-])=O)S(=O)(=O)Nc1cc(Cl)ccc1S(C)=O
Show InChI InChI=1S/C14H13ClN2O5S2/c1-9-3-5-11(8-13(9)17(18)19)24(21,22)16-12-7-10(15)4-6-14(12)23(2)20/h3-8,16H,1-2H3
PDB

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n/an/a 181n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327275
PNG
(4-chloro-N-{5-chloro-2-[(1H-imidazol-2-ylmethyl)th...)
Show SMILES FC(F)(F)c1cc(ccc1Cl)S(=O)(=O)Nc1cc(Cl)ccc1SCc1ncc[nH]1
Show InChI InChI=1S/C17H12Cl2F3N3O2S2/c18-10-1-4-15(28-9-16-23-5-6-24-16)14(7-10)25-29(26,27)11-2-3-13(19)12(8-11)17(20,21)22/h1-8,25H,9H2,(H,23,24)
PDB

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n/an/a 190n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327237
PNG
(4-chloro-N-[5-chloro-2-(ethylthio)phenyl]-3-(trifl...)
Show SMILES CCSc1ccc(Cl)cc1NS(=O)(=O)c1ccc(Cl)c(c1)C(F)(F)F
Show InChI InChI=1S/C15H12Cl2F3NO2S2/c1-2-24-14-6-3-9(16)7-13(14)21-25(22,23)10-4-5-12(17)11(8-10)15(18,19)20/h3-8,21H,2H2,1H3
PDB

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UniProtKB/SwissProt

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PC cid
PC sid
UniChem
US Patent
n/an/a 193n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327263
PNG
(N-[5-chloro-2-(methylsulfinyl)phenyl]-5-methylfura...)
Show SMILES Cc1ccc(o1)S(=O)(=O)Nc1cc(Cl)ccc1S(C)=O
Show InChI InChI=1S/C12H12ClNO4S2/c1-8-3-6-12(18-8)20(16,17)14-10-7-9(13)4-5-11(10)19(2)15/h3-7,14H,1-2H3
PDB

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UniProtKB/SwissProt

GoogleScholar
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PC cid
PC sid
UniChem
US Patent
n/an/a 194n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327366
PNG
(N-{5-chloro-2-[(2-pyridin-2-ylethyl)sulfonyl]-phen...)
Show SMILES Clc1ccc(c(NS(=O)(=O)c2cc3ccccc3o2)c1)S(=O)(=O)CCc1ccccn1
Show InChI InChI=1S/C21H17ClN2O5S2/c22-16-8-9-20(30(25,26)12-10-17-6-3-4-11-23-17)18(14-16)24-31(27,28)21-13-15-5-1-2-7-19(15)29-21/h1-9,11,13-14,24H,10,12H2
PDB

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UniProtKB/SwissProt

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PC cid
PC sid
UniChem
US Patent
n/an/a 197n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327222
PNG
(4-chloro-N-{5-chloro-2-[(pyridin-2-ylmethyl)thio]-...)
Show SMILES FC(F)(F)c1cc(ccc1Cl)S(=O)(=O)Nc1cc(Cl)ccc1SCc1ccccn1
Show InChI InChI=1S/C19H13Cl2F3N2O2S2/c20-12-4-7-18(29-11-13-3-1-2-8-25-13)17(9-12)26-30(27,28)14-5-6-16(21)15(10-14)19(22,23)24/h1-10,26H,11H2
PDB

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UniProtKB/SwissProt

GoogleScholar
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PC cid
PC sid
UniChem
US Patent
n/an/a 199n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327247
PNG
(N-[5-chloro-2-(methylsulfonyl)phenyl]-4-methyl-3-n...)
Show SMILES Cc1ccc(cc1[N+]([O-])=O)S(=O)(=O)Nc1cc(Cl)ccc1S(C)(=O)=O
Show InChI InChI=1S/C14H13ClN2O6S2/c1-9-3-5-11(8-13(9)17(18)19)25(22,23)16-12-7-10(15)4-6-14(12)24(2,20)21/h3-8,16H,1-2H3
PDB

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UniProtKB/SwissProt

GoogleScholar
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PC cid
PC sid
UniChem
US Patent
n/an/a 207n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
C-C chemokine receptor type 2


(Homo sapiens (Human))
BDBM327362
PNG
(3-[(4-chloro-2-{[(4-chloro-2-fluorophenyl)sulfonyl...)
Show SMILES CN(C)C(=O)CCS(=O)(=O)c1ccc(Cl)cc1NS(=O)(=O)c1ccc(Cl)cc1F
Show InChI InChI=1S/C17H17Cl2FN2O5S2/c1-22(2)17(23)7-8-28(24,25)16-6-4-12(19)10-14(16)21-29(26,27)15-5-3-11(18)9-13(15)20/h3-6,9-10,21H,7-8H2,1-2H3
PDB

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UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 211n/an/an/an/an/an/a



ALLERGAN, INC.

US Patent


Assay Description
HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...


US Patent US9663460 (2017)

More data for this
Ligand-Target Pair
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* indicates data uncertainty>20%