Compile Data Set for Download or QSAR
maximum 50k data
Found 125 Enz. Inhib. hit(s) with all data for entry = 1525
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329844((rac)-((1R,2R,3S,4R)-4-(2-(6-tert-butylpyridin-2-y...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329845((rac)-((1R,2R,3S,4R)-4-(2-(3,3-dimethyl-1,3-dihydr...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329846((rac)-[(1R,2R,3S,4R)-4-{[2-(5-chloro-1H-indol-3-yl...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329847((rac)-[(1R,2R,3S,4R)-4-{[2-(6-chloro-1H-indol-3-yl...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329848((rac)-((1R,2R,3S,4R)-4-((2-(Dibenzo[b,d]thiophen-4...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329849((rac)-((1R,2R,3S,4R)-4-(2-(5-chloro-2-(trifluorome...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329850((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(1,1,1-...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329853((rac)-((1R,2R,3S,4R)-4-((2-(Benzo[b]thiophen-4-yl)...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329854((rac)-[(1R,2R,3S,4R)-4-{[2-(9H-carbazol-2-yl)pyraz...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329807((rac)-((1R,2R,3S,4R)-4-((2-(3-(tert-Butyl)phenyl)p...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329857((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(2-methox...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329858((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(2-methox...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329859((rac)-[(1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(2-phenyl...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329862((rac)-((1R,2R,3S,4R)-4-(2-(4-fluoro-2-methoxypheny...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329863((rac)-((1R,2R,3S,4R)-4-(2-(5-chlorobenzo[b]thiophe...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329864((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-methoyp...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329867((rac)-((1R,2R,3S,4R)-4-(2-(1H-indol-4-yl)pyrazolo[...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329868((rac)-((1R,2R,3S,4R)-4-(2-(3-(cyclopropylmethylthi...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329869((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(piperi...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329870((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-morphol...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329873((rac)-((1R,2R,3S,4R)-4-(2-(5-fluorobenzo[b]thiophe...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329874((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(2-meth...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329875((rac)-[(1R,2R,3S,4R)-4-{[2-(3-ethynylphenyl)pyrazo...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329876((rac)-((1R,2R,3S,4R)-4-(2-(3-(2-ethoxypropan-2-yl)...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329877((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(9-oxo-9H-...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329878((rac)-((1R,2R,3S,4R)-4-(2-(benzofuran-2-yl)pyrazol...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329879((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(2-oxop...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329882((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(2-prop...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329883((rac)-((1R,2R,3S,4R)-4-(2-(6-chlorobenzo[b]thiophe...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329884((rac)-((1R,2R,3S,4R)-4-(2-(5-chlorobenzofuran-3-yl...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329885((rac)-((1R,2R,3S,4R)-4-(2-(dibenzo[b,d]furan-3-yl)...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329886((rac)-((1R,2R,3S,4R)-4-(2-(5-ethylbenzo[b]thiophen...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329888((rac)-methyl rel-5-[7-({(1R,2S,3R,4R)-2,3-dihydrox...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329889((rac)-((1R,2R,3S,4R)-4-(2-(5-fluoronaphthalen-1-yl...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329794((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(1-naphth...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329891((rac)-rel-5-[7-({(1R,2S,3R,4R)-2,3-dihydroxy-4- | ...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329892((s.e.)-((1R,2R,3S,4R)-4-(2-(4-fluoronaphthalen-1-y...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329836((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(triflu...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329858((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(2-methox...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329802((rac)-((1R,2R,3S,4R)-4-(2-(dibenzo[b,d]furan-4-yl)...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329896((s.e.)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-methox...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329889((rac)-((1R,2R,3S,4R)-4-(2-(5-fluoronaphthalen-1-yl...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329898((s.e.)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(4-methox...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329899((s.e.)-((1R,2R,3S,4R)-4-(2-(4-(dimethylamino)napht...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329900((s.e.)-[(1R,2R,3S,4R)-4-{[2-(4-chloro-1-naphthyl)p...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329901((s.e.)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-isopro...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329902((s.e.)-((1R,2R,3S,4R)-4-(2-(2-(difluoromethoxy)nap...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329903((s.e.)-((1R,2R,3S,4R)-4-(2-(6-(difluoromethyl)naph...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329904((s.e.)-((1R,2R,3S,4R)-4-(2-(4-(difluoromethoxy)nap...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin-conjugating enzyme E2 E1(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329905((s.e.)-((1R,2R,3S,4R)-4-(2-(6-fluoronaphthalen-2-y...)
Affinity DataIC50: <10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 125 total ) | Next | Last >>
Jump to: