Affinity Data by Patent

Patent code US9663525

Found 125 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329807 ((rac)-((1R,2R,3S,4R)-4-((2-(3-(tert-Butyl)phenyl)p...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329863 ((rac)-((1R,2R,3S,4R)-4-(2-(5-chlorobenzo[b]thiophe...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329886 ((rac)-((1R,2R,3S,4R)-4-(2-(5-ethylbenzo[b]thiophen...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329888 ((rac)-methyl rel-5-[7-({(1R,2S,3R,4R)-2,3-dihydrox...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329892 ((s.e.)-((1R,2R,3S,4R)-4-(2-(4-fluoronaphthalen-1-y...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329836 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(triflu...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329802 ((rac)-((1R,2R,3S,4R)-4-(2-(dibenzo[b,d]furan-4-yl)...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329902 ((s.e.)-((1R,2R,3S,4R)-4-(2-(2-(difluoromethoxy)nap...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329914 ((rac)-[(1R,2R,3S,4R)-2,3-dihydroxy-4-({2-[3-(1-met...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329802 ((rac)-((1R,2R,3S,4R)-4-(2-(dibenzo[b,d]furan-4-yl)...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329808 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(naphthale...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329811 ((rac)-((1R,2R,3S,4R)-4-(2-(dibenzo[b,d]furan-2-yl)...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329812 ((rac)-((1R,2R,3S,4R)-4-(2-(5-chloro-2-methoxypheny...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329816 ((rac)-((1R,2R,3S,4R)-4-(2-(1H-indol-2-yl)pyrazolo[...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329828 ((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(3-(pyrid...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329830 ((rac)-[(1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(5-methyl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329849 ((rac)-((1R,2R,3S,4R)-4-(2-(5-chloro-2-(trifluorome...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329875 ((rac)-[(1R,2R,3S,4R)-4-{[2-(3-ethynylphenyl)pyrazo...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329879 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(2-oxop...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329885 ((rac)-((1R,2R,3S,4R)-4-(2-(dibenzo[b,d]furan-3-yl)...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329901 ((s.e.)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-isopro...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329904 ((s.e.)-((1R,2R,3S,4R)-4-(2-(4-(difluoromethoxy)nap...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329905 ((s.e.)-((1R,2R,3S,4R)-4-(2-(6-fluoronaphthalen-2-y...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329906 ((s.e.)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-methyl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329824 ((rac)-[(1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(1H-indol...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329839 ((rac)-(1R,2R,3S,4R)-4-(2-(3-cyclopentenylphenyl)py...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329840 ((rac)-[(1R,2R,3S,4R)-4-{[2-(3-cyclopentylphenyl)py...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329841 ((rac)-((1R,2R,3S,4R)-4-(2-(benzofuran-3-yl)pyrazol...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329844 ((rac)-((1R,2R,3S,4R)-4-(2-(6-tert-butylpyridin-2-y...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329853 ((rac)-((1R,2R,3S,4R)-4-((2-(Benzo[b]thiophen-4-yl)...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329818 ((rac)-((1R,2R,3S,4R)-4-(2-(3,3-dimethyl-2,3-dihydr...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329827 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(trimet...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329833 ((rac)-((1R,2R,3S,4R)-4-(2-(3,3-dimethyl-2,3-dihydr...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329837 ((rac)-((1R,2R,3S,4R)-4-((2-(Benzo[b]thiophen-7-yl)...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329846 ((rac)-[(1R,2R,3S,4R)-4-{[2-(5-chloro-1H-indol-3-yl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329873 ((rac)-((1R,2R,3S,4R)-4-(2-(5-fluorobenzo[b]thiophe...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329877 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(9-oxo-9H-...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329878 ((rac)-((1R,2R,3S,4R)-4-(2-(benzofuran-2-yl)pyrazol...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329883 ((rac)-((1R,2R,3S,4R)-4-(2-(6-chlorobenzo[b]thiophe...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329889 ((rac)-((1R,2R,3S,4R)-4-(2-(5-fluoronaphthalen-1-yl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329900 ((s.e.)-[(1R,2R,3S,4R)-4-{[2-(4-chloro-1-naphthyl)p...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329813 ((rac)-((1R,2R,3S,4R)-4-(2-(5-chloro-2-methylphenyl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329826 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(quinolin-...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329832 ((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(3-(trifl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329845 ((rac)-((1R,2R,3S,4R)-4-(2-(3,3-dimethyl-1,3-dihydr...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329858 ((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(2-methox...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329868 ((rac)-((1R,2R,3S,4R)-4-(2-(3-(cyclopropylmethylthi...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329876 ((rac)-((1R,2R,3S,4R)-4-(2-(3-(2-ethoxypropan-2-yl)...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329882 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(2-prop...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329884 ((rac)-((1R,2R,3S,4R)-4-(2-(5-chlorobenzofuran-3-yl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329896 ((s.e.)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-methox...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329898 ((s.e.)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(4-methox...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329899 ((s.e.)-((1R,2R,3S,4R)-4-(2-(4-(dimethylamino)napht...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329907 ((s.e.)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(4-methyl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329911 ((s.e.)-((1R,2R,3S,4R)-4-(2-(1-fluoronaphthalen-2-y...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329819 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(isoquinol...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329825 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(5-(triflu...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329835 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(quinolin-...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329836 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(triflu...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329848 ((rac)-((1R,2R,3S,4R)-4-((2-(Dibenzo[b,d]thiophen-4...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329857 ((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(2-methox...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329859 ((rac)-[(1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(2-phenyl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329869 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(piperi...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329870 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-morphol...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329874 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(2-meth...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329858 ((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(2-methox...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329908 ((s.e.)-((1R,2R,3S,4R)-4-(2-(3-fluoronaphthalen-2-y...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329913 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(6-phenyl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329915 ((rac)-{(1R,2R,3S,4R)-4-[(2-{3-[2-chloro-1-(hydroxy...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329794 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(1-naphth...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329799 ((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(3-(trifl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329807 ((rac)-((1R,2R,3S,4R)-4-((2-(3-(tert-Butyl)phenyl)p...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329809 ((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(quinolin...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329814 ((rac)-((1R,2R,3S,4R)-4-(2-(benzo[b]thiophen-3-yl)p...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329822 ((rac)-((1R,2R,3S,4R)-4-((2-(2-Chloro-5-(trifluorom...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329823 ((rac)-[(1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(4-phenyl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329834 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(quinolin-...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329838 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(pyrrol...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329842 ((rac)-((1R,2R,3S,4R)-4-((2-(3-(Difluoromethoxy)phe...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329850 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(1,1,1-...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329862 ((rac)-((1R,2R,3S,4R)-4-(2-(4-fluoro-2-methoxypheny...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329867 ((rac)-((1R,2R,3S,4R)-4-(2-(1H-indol-4-yl)pyrazolo[...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329889 ((rac)-((1R,2R,3S,4R)-4-(2-(5-fluoronaphthalen-1-yl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329903 ((s.e.)-((1R,2R,3S,4R)-4-(2-(6-(difluoromethyl)naph...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329795 ((rac)((1R,2R,3S,4R)-4-(2-(biphenyl-3-yl)pyrazolo[1...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329820 ((rac)-((1R,2R,3S,4R)-4-((2-(3-Bromophenyl)pyrazolo...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329821 ((rac)-((1R,2R,3S,4R)-4-((2-(2-Fluoro-5-(trifluorom...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329831 ((rac)-((1R,2R,3S,4R)-4-(2-(7-chloroquinolin-4-yl)p...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329847 ((rac)-[(1R,2R,3S,4R)-4-{[2-(6-chloro-1H-indol-3-yl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329854 ((rac)-[(1R,2R,3S,4R)-4-{[2-(9H-carbazol-2-yl)pyraz...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329864 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-methoyp...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329794 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(1-naphth...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329891 ((rac)-rel-5-[7-({(1R,2S,3R,4R)-2,3-dihydroxy-4- \| ...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329910 ((s.e.)-((1R,2R,3S,4R)-4-(2-(4-fluoronaphthalen-2-y...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329912 ((s.e.)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-methox...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329797 ((rac)-((1R,2R,3S,4R)-4-((2-(3-Chlorophenyl)pyrazol...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329810 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(isoquinol...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329829 ((rac)-[(1R,2R,3S,4R)-4-{[2-(9H-carbazol-3-yl)pyraz...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329843 ((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(3-phenox...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329852 ((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(5-(trifl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329861 ((rac)-((1R,2R,3S,4R)-4-(2-(3-benzylpenyl)pyrazolo[...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329805 ((rac)-[(1R,2R,3S,4R)-4-{[2-(2,4-dichlorophenyl)pyr...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329872 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(4-(triflu...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329880 ((rac)-((1R,2R,3S,4R)-4-(2-(6-chlorobenzo[b]thiophe...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329871 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-(triflu...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329856 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(6-(triflu...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329851 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-(triflu...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329793 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-phenylpyra...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329866 ((rac)-[(1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(1H-indol...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329860 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-phenoxy...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329804 ((rac)-[(1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(pyridin-...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329815 ((rac)-((1R,2R,3S,4R)-4-(2-(3,3-dimethyl-2,3-dihydr...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329865 ((rac)-((1R,2R,3S,4R)-4-(2-(3-benzoylphenyl)pyrazol...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329909 ((s.e.)-((1R,2R,3S,4R)-4-(2-(2,4-dichloronaphthalen...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329817 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(quinolin-...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329887 ((rac)-((1R,2R,3S,4R)-4-(2-(5-ethylbenzo[b]thiophen...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329916 ((s.e.)-{(1R,2R,3S,4R)-4-[(3,6-dichloro-2-{3- \| US9...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329917 ((s.e.)-{(1R,2R,3S,4R)-4-[(6-chloro-2-{3-[(trifluor...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329803 ((rac)-((1R,2R,3S,4R)-4-(5-chloro-2-(pyridin-2-yl)p...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329806 ((rac)-[(1R,2R,3S,4R)-4-{[5-chloro-2-(4-methoxyphen...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329801 ((rac)-((1R,2R,3S,4R)-4-{[5-chloro-2-(1-naphthyl)py...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329800 ((rac)-((1R,2R,3S,4R)-4-(2-(4-bromophenyl)-5-chloro...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329881 ((rac)-{(1R,2R,3S,4R)-2,3-dihydroxy-4-[(6-methyl-2-...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329798 ((rac)-{(1R,2R,3S,4R)-4-[(5-chloro-2-phenylpyrazolo...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair
E2 ubiquitin-conjugating enzyme E1 (Homo sapiens (Human))	BDBM329796 ((rac)-{(1R,2R,3S,4R)-2,3-dihydroxy-4-[(5-methyl-2-...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	n/a
Millennium Pharmaceuticals, Inc. US Patent					Assay Description The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...				US Patent US9663525 (2017)
Millennium Pharmaceuticals, Inc. US Patent					More data for this Ligand-Target Pair