Compile Data Set for Download or QSAR
maximum 50k data
Found 150 Enz. Inhib. hit(s) with all data for entry = 103
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174126(US9688668, 1a)
Affinity DataKi:  100nMAssay Description:SLR080811, prepared as the HCl salt, was tested first at recombinant SphK1 and SphK2 using a broken cell assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174047(US9688668, 15)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174049(US9688668, 16)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174050(US9688668, 17)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174053(US9688668, 20)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174054(US9688668, 21)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174055(US9688668, 22)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174056(US9688668, 23)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174059(US9688668, 24)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174060(US9688668, 25)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174061(US9688668, 26)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174063(US9688668, 27)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174064(US9688668, 28)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174065(US9688668, 29)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174066(US9688668, 30)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174067(US9688668, 31)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174068(US9688668, 32)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174114(US9688668, 64)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174044(US9688668, 13)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174046(US9688668, 14)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM50443388(CHEMBL3086782 | US9688668, SLR080811)
Affinity DataKi:  1.30E+3nMAssay Description:SLR080811, prepared as the HCl salt, was tested first at recombinant SphK1 and SphK2 using a broken cell assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174126(US9688668, 1a)
Affinity DataKi:  1.50E+3nMAssay Description:SLR080811, prepared as the HCl salt, was tested first at recombinant SphK1 and SphK2 using a broken cell assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174009(US9688668, 1)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174009(US9688668, 1)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174010(US9688668, 2)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174010(US9688668, 2)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174022(US9688668, 4)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174022(US9688668, 4)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174023(US9688668, 5)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174023(US9688668, 5)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174026(US9688668, 6)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174026(US9688668, 6)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174028(US9688668, 7)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174028(US9688668, 7)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174038(US9688668, 8)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174038(US9688668, 8)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174043(US9688668, 12)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174043(US9688668, 12)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174049(US9688668, 16)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174051(US9688668, 18)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174051(US9688668, 18)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174052(US9688668, 19)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174052(US9688668, 19)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174069(US9688668, 33)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174069(US9688668, 33)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174070(US9688668, 34)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174071(US9688668, 35)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174071(US9688668, 35)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174072(US9688668, 36)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia Patent Foundation

US Patent
LigandPNGBDBM174072(US9688668, 36)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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