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Found 46 Enz. Inhib. hit(s) with all data for entry = 114
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM235683(Estradiol-17β (3) | US9688816, A)
Affinity DataIC50:  1nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM235683(Estradiol-17β (3) | US9688816, A)
Affinity DataIC50:  6.60nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM235683(Estradiol-17β (3) | US9688816, A)
Affinity DataIC50:  7nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM235683(Estradiol-17β (3) | US9688816, A)
Affinity DataIC50:  8.20nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM235683(Estradiol-17β (3) | US9688816, A)
Affinity DataIC50:  10nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM235683(Estradiol-17β (3) | US9688816, A)
Affinity DataIC50:  15nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176759(CAS# 129188-99-4 | Hydro Isophorone Bisphenol | US...)
Affinity DataIC50:  450nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM29608(Bisphenol A (BPA) | Diphenylolpropane | US9688816,...)
Affinity DataIC50:  490nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM29608(Bisphenol A (BPA) | Diphenylolpropane | US9688816,...)
Affinity DataIC50:  670nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176759(CAS# 129188-99-4 | Hydro Isophorone Bisphenol | US...)
Affinity DataIC50:  1.10E+3nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176753(CAS# 2362-14-3 | Dimethyl Cyclohexyl Bisphenol | U...)
Affinity DataIC50:  1.30E+3nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176760(Bisphenol M | CAS# 13595-25-0 | US9688816, K)
Affinity DataIC50:  1.40E+3nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM29337(US9688816, D | triphenylmethane derivative, 9)
Affinity DataIC50:  1.40E+3nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM50121958(4,4'-Biphenyldiol | 4,4'-Dihydroxybiphenyl | 4,4'-...)
Affinity DataIC50:  1.70E+3nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176760(Bisphenol M | CAS# 13595-25-0 | US9688816, K)
Affinity DataIC50:  2.10E+3nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176753(CAS# 2362-14-3 | Dimethyl Cyclohexyl Bisphenol | U...)
Affinity DataIC50:  3.10E+3nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176750(CAS# 4754-63-6 | Dimethyl Acetophenone Bisphenol |...)
Affinity DataIC50:  3.50E+3nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM50077844(3,3-Bis-(4-hydroxy-phenyl)-3H-isobenzofuran-1-one ...)
Affinity DataIC50:  3.70E+3nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176750(CAS# 4754-63-6 | Dimethyl Acetophenone Bisphenol |...)
Affinity DataIC50:  4.80E+3nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176758(CAS# 88938-12-9 | Fluorenone Bis-o-Cresol | US9688...)
Affinity DataIC50:  9.70E+3nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM29609(4-alpha-Cumylphenol | 4-cumylphenol | US9688816, B)
Affinity DataIC50:  9.80E+3nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176752(CAS# 7297-85-0 | Diphenolic Acid Methyl Ester | US...)
Affinity DataIC50:  1.10E+4nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM29337(US9688816, D | triphenylmethane derivative, 9)
Affinity DataIC50:  1.20E+4nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM76095(4-(4-hydroxyphenoxy)phenol | 4-(4-oxidanylphenoxy)...)
Affinity DataIC50:  1.40E+4nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM50077844(3,3-Bis-(4-hydroxy-phenyl)-3H-isobenzofuran-1-one ...)
Affinity DataIC50:  1.40E+4nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176752(CAS# 7297-85-0 | Diphenolic Acid Methyl Ester | US...)
Affinity DataIC50:  1.90E+4nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176758(CAS# 88938-12-9 | Fluorenone Bis-o-Cresol | US9688...)
Affinity DataIC50:  2.50E+4nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM25807(4,4 -Dihydroxybenzophenone | 4-[(4-hydroxyphenyl)c...)
Affinity DataIC50:  3.10E+4nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM25807(4,4 -Dihydroxybenzophenone | 4-[(4-hydroxyphenyl)c...)
Affinity DataIC50:  3.20E+4nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM76095(4-(4-hydroxyphenoxy)phenol | 4-(4-oxidanylphenoxy)...)
Affinity DataIC50:  6.00E+4nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM29609(4-alpha-Cumylphenol | 4-cumylphenol | US9688816, B)
Affinity DataIC50:  1.40E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176762(CAS# 1568-80-5 | Spiro Biindane Bisphenol | US9688...)
Affinity DataIC50: >2.50E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176762(CAS# 1568-80-5 | Spiro Biindane Bisphenol | US9688...)
Affinity DataIC50: >2.50E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM50121958(4,4'-Biphenyldiol | 4,4'-Dihydroxybiphenyl | 4,4'-...)
Affinity DataIC50: >2.50E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM34126(US9688816, 1 | bis(2,6-dimethylphenol), 2)
Affinity DataIC50: >2.50E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176764(2,5-Di-tert-butylhydroquinone | CAS# 88-58-4 | US9...)
Affinity DataIC50: >2.50E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176764(2,5-Di-tert-butylhydroquinone | CAS# 88-58-4 | US9...)
Affinity DataIC50: >2.50E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM34126(US9688816, 1 | bis(2,6-dimethylphenol), 2)
Affinity DataIC50: >2.50E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176768(CAS# 95-71-6 | Methyl Hydroquinone | US9688816, 8)
Affinity DataIC50: >2.50E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM26187(α-CA inhibitor, 11 | CHEMBL14060 | US9688816,...)
Affinity DataIC50: >2.50E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM26187(α-CA inhibitor, 11 | CHEMBL14060 | US9688816,...)
Affinity DataIC50: >2.50E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176756(CAS# 6607-41-6 | N-Phenyl Phenolphthalein Bispheno...)
Affinity DataIC50: >2.50E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176756(CAS# 6607-41-6 | N-Phenyl Phenolphthalein Bispheno...)
Affinity DataIC50: >2.50E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM26189(α-CA inhibitor, 13 | 1,3-Dihydroxybenzene, XI...)
Affinity DataIC50: >2.50E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM176768(CAS# 95-71-6 | Methyl Hydroquinone | US9688816, 8)
Affinity DataIC50: >2.50E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor beta(Homo sapiens (Human))
Sabic Global Technologies

US Patent
LigandPNGBDBM26189(α-CA inhibitor, 13 | 1,3-Dihydroxybenzene, XI...)
Affinity DataIC50: >2.50E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent