Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 28
TargetEpidermal growth factor receptor [L858R](Homo sapiens (Human))
Jiangsu Medolution

US Patent
LigandPNGBDBM76963(US9694011, Example 1 (Compound 17))
Affinity DataKd:  54nMT: 2°CAssay Description:Kinase-tagged T7 phage strains were prepared in an E. coli host derived from the BL21 strain. E. coli were grown to log-phase and infected with T7 ph...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEpidermal growth factor receptor [L858R](Homo sapiens (Human))
Jiangsu Medolution

US Patent
LigandPNGBDBM76973(US9694011, Example 2 (Compound 18))
Affinity DataKd:  6.30nMT: 2°CAssay Description:Kinase-tagged T7 phage strains were prepared in an E. coli host derived from the BL21 strain. E. coli were grown to log-phase and infected with T7 ph...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Medolution

US Patent
LigandPNGBDBM76973(US9694011, Example 2 (Compound 18))
Affinity DataKd: <10nMT: 2°CAssay Description:Kinase-tagged T7 phage strains were prepared in an E. coli host derived from the BL21 strain. E. coli were grown to log-phase and infected with T7 ph...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEpidermal growth factor receptor [T790M,L858R](Homo sapiens (Human))
Jiangsu Medolution

US Patent
LigandPNGBDBM76973(US9694011, Example 2 (Compound 18))
Affinity DataKd:  9.30nMT: 2°CAssay Description:Kinase-tagged T7 phage strains were prepared in an E. coli host derived from the BL21 strain. E. coli were grown to log-phase and infected with T7 ph...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Medolution

US Patent
LigandPNGBDBM76963(US9694011, Example 1 (Compound 17))
Affinity DataKd: <10nMT: 2°CAssay Description:Kinase-tagged T7 phage strains were prepared in an E. coli host derived from the BL21 strain. E. coli were grown to log-phase and infected with T7 ph...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEpidermal growth factor receptor [T790M,L858R](Homo sapiens (Human))
Jiangsu Medolution

US Patent
LigandPNGBDBM76963(US9694011, Example 1 (Compound 17))
Affinity DataKd:  270nMT: 2°CAssay Description:Kinase-tagged T7 phage strains were prepared in an E. coli host derived from the BL21 strain. E. coli were grown to log-phase and infected with T7 ph...More data for this Ligand-Target Pair
In DepthDetails US Patent