Compile Data Set for Download or QSAR
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Found 8 Enz. Inhib. hit(s) with all data for entry = 1643
TargetAndrogen receptor(Homo sapiens (Human))
Galderma Research & Development

US Patent
LigandPNGBDBM334271(2-Hydroxy-2- methyl- pentanoic acid (2-bromo-pyrid...)
Affinity DataKd:  75nMAssay Description:The N-(pyrid-4-yl)amides and N-(pyrimidin-4-yl)amides described herein exhibit androgen receptor (AR) inhibiting properties. This AR inhibiting activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Galderma Research & Development

US Patent
LigandPNGBDBM334272(2-Hydroxy-2- methyl-hexanoic acid (2-bromo- 6-meth...)
Affinity DataKd:  30nMAssay Description:The N-(pyrid-4-yl)amides and N-(pyrimidin-4-yl)amides described herein exhibit androgen receptor (AR) inhibiting properties. This AR inhibiting activ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Galderma Research & Development

US Patent
LigandPNGBDBM334273(2-Butyl-2- hydroxy-hexanoic acid (2-bromo- pyridin...)
Affinity DataKd:  15nMAssay Description:The N-(pyrid-4-yl)amides and N-(pyrimidin-4-yl)amides described herein exhibit androgen receptor (AR) inhibiting properties. This AR inhibiting activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Galderma Research & Development

US Patent
LigandPNGBDBM334278(4-(2-Hydroxy-2- methyl- pentanoylamino)- pyridine-...)
Affinity DataKd:  6.00E+3nMAssay Description:The N-(pyrid-4-yl)amides and N-(pyrimidin-4-yl)amides described herein exhibit androgen receptor (AR) inhibiting properties. This AR inhibiting activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Galderma Research & Development

US Patent
LigandPNGBDBM334275(N-(2-Bromo- pyridin-4-yl)-2- hydroxy-2-phenyl- pro...)
Affinity DataKd:  100nMAssay Description:The N-(pyrid-4-yl)amides and N-(pyrimidin-4-yl)amides described herein exhibit androgen receptor (AR) inhibiting properties. This AR inhibiting activ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Galderma Research & Development

US Patent
LigandPNGBDBM334276(2-Hydroxy-2,4- dimethyl-pentanoic acid (2-bromo-6-...)
Affinity DataKd:  20nMAssay Description:The N-(pyrid-4-yl)amides and N-(pyrimidin-4-yl)amides described herein exhibit androgen receptor (AR) inhibiting properties. This AR inhibiting activ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Galderma Research & Development

US Patent
LigandPNGBDBM334277(N-(2-Bromo-pyridin- 4-yl)-2-hydroxy- 2-methyl-4-ph...)
Affinity DataKd:  100nMAssay Description:The N-(pyrid-4-yl)amides and N-(pyrimidin-4-yl)amides described herein exhibit androgen receptor (AR) inhibiting properties. This AR inhibiting activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Galderma Research & Development

US Patent
LigandPNGBDBM334274(N-(2-Bromo-pyridin- 4-yl)-2-hydroxy-4- (4-methoxy-...)
Affinity DataKd:  300nMAssay Description:The N-(pyrid-4-yl)amides and N-(pyrimidin-4-yl)amides described herein exhibit androgen receptor (AR) inhibiting properties. This AR inhibiting activ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent