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Patent code US9737516

Compile Data Set for Download or QSAR
Found 44 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333406
PNG
(6-(2,4-Difluorophenoxy)-1-methyl-5-(6-methyl-7-oxo...)
Show SMILES Cn1c2cc(Oc3ccc(F)cc3F)c(cc2[nH]c1=O)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C17H16Cl2N4O2S/c18-10-3-1-2-9(4-10)5-20-16-17-21-6-11(23(17)7-13(19)22-16)15-14(25)12(24)8-26-15/h1-4,6-7,12,14-15,24-25H,5,8H2,(H,20,22)/t12-,14-,15+/m1/s1
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UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333424
PNG
(4-[5-(Cyclobutylmethoxy)-2-piperidin-1-yl-1H-benzi...)
Show SMILES Cn1cc(-c2cc3[nH]c(nc3cc2OCC2CCC2)N2CCCCC2)c2cc[nH]c2c1=O
Show InChI InChI=1S/C17H17ClFN5O2/c18-10-1-3-12(19)9(7-10)8-21-15-17-23-22-16(24(17)6-5-20-15)11-2-4-13(25)14(11)26/h1,3,5-7,11,13-14,25-26H,2,4,8H2,(H,20,21)/t11-,13-,14+/m1/s1
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UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333414
PNG
(4-[6-(2,4-Difluorophenoxy)-1,3-dimethyl-2-oxo-2,3-...)
Show SMILES Cn1c2cc(Oc3ccc(F)cc3F)c(cc2n(C)c1=O)-c1cn(C)c(=O)c2[nH]ncc12
Show InChI InChI=1S/C18H18ClFN4O2/c19-11-1-3-13(20)10(7-11)8-22-17-18-23-9-14(24(18)6-5-21-17)12-2-4-15(25)16(12)26/h1,3,5-7,9,12,15-16,25-26H,2,4,8H2,(H,21,22)/t12-,15+,16-/m0/s1
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UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333422
PNG
(4-[5-(Cyclobutylmethoxy)-1-isopropyl-1H-benzimidaz...)
Show SMILES CC(C)n1cnc2cc(OCC3CCC3)c(cc12)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C17H17Cl2N5O2/c18-10-5-9(6-11(19)7-10)8-21-15-17-23-22-16(24(17)4-3-20-15)12-1-2-13(25)14(12)26/h3-7,12-14,25-26H,1-2,8H2,(H,20,21)/t12-,13-,14+/m1/s1
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UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333409
PNG
(4-[5-(2,4-Difluorophenoxy)-1H-benzimidazol-6-yl]-6...)
Show SMILES Cn1cc(-c2cc3[nH]cnc3cc2Oc2ccc(F)cc2F)c2cc[nH]c2c1=O
Show InChI InChI=1S/C18H17Cl2N3O2S/c19-11-3-1-2-10(4-11)6-21-13-5-12(20)8-23-14(7-22-18(13)23)17-16(25)15(24)9-26-17/h1-5,7-8,15-17,21,24-25H,6,9H2/t15-,16-,17+/m1/s1
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UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333412
PNG
(4-(5-(2,4-difluorophenoxy)-1H-benzo[d][1,2,3]triaz...)
Show SMILES Cn1cc(-c2cc3[nH]nnc3cc2Oc2ccc(F)cc2F)c2cc[nH]c2c1=O
Show InChI InChI=1S/C18H18Cl2N4O2/c19-11-5-10(6-12(20)7-11)8-22-17-18-23-9-14(24(18)4-3-21-17)13-1-2-15(25)16(13)26/h3-7,9,13,15-16,25-26H,1-2,8H2,(H,21,22)/t13-,15+,16-/m0/s1
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UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333413
PNG
(4-[6-(2,4-Difluorophenoxy)-1H-benzimidazol-5-yl]-6...)
Show SMILES Cn1cc(-c2cc3[nH]cnc3cc2Oc2ccc(F)cc2F)c2cn[nH]c2c1=O
Show InChI InChI=1S/C18H18Cl2N4O2/c19-11-1-3-13(20)10(7-11)8-22-17-18-23-9-14(24(18)6-5-21-17)12-2-4-15(25)16(12)26/h1,3,5-7,9,12,15-16,25-26H,2,4,8H2,(H,21,22)/t12-,15+,16-/m0/s1
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PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333415
PNG
(4-[5-(Cyclobutylmethoxy)-1H-benzimidazol-6-yl]-6-m...)
Show SMILES Cn1cc(-c2cc3NCNc3cc2OCC2CCC2)c2cc[nH]c2c1=O
Show InChI InChI=1S/C19H21FN4O2/c20-13-3-1-12(2-4-13)7-8-21-18-19-23-11-15(24(19)10-9-22-18)14-5-6-16(25)17(14)26/h1-4,9-11,14,16-17,25-26H,5-8H2,(H,21,22)/t14-,16+,17-/m0/s1
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PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333418
PNG
(4-[5-(Cyclobutylmethoxy)-1-methyl-1H-benzimidazol-...)
Show SMILES Cn1cnc2cc(OCC3CCC3)c(cc12)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C19H20ClFN4O2/c20-13-9-11(1-3-14(13)21)5-6-22-18-19-24-10-15(25(19)8-7-23-18)12-2-4-16(26)17(12)27/h1,3,7-10,12,16-17,26-27H,2,4-6H2,(H,22,23)/t12-,16+,17-/m0/s1
GoogleScholar
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PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333405
PNG
(5-(2,4-Difluorophenoxy)-6-(6-methyl-7-oxo-6,7-dihy...)
Show SMILES Cn1cc(-c2cc3[nH]c(=O)[nH]c3cc2Oc2ccc(F)cc2F)c2cc[nH]c2c1=O
Show InChI InChI=1S/C19H19ClN4O2S/c20-11-3-1-2-10(6-11)12-7-13(12)23-18-19-22-8-14(24(19)5-4-21-18)17-16(26)15(25)9-27-17/h1-6,8,12-13,15-17,25-26H,7,9H2,(H,21,23)/t12-,13+,15-,16-,17+/m1/s1
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UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333414
PNG
(4-[6-(2,4-Difluorophenoxy)-1,3-dimethyl-2-oxo-2,3-...)
Show SMILES Cn1c2cc(Oc3ccc(F)cc3F)c(cc2n(C)c1=O)-c1cn(C)c(=O)c2[nH]ncc12
Show InChI InChI=1S/C18H18ClFN4O2/c19-11-1-3-13(20)10(7-11)8-22-17-18-23-9-14(24(18)6-5-21-17)12-2-4-15(25)16(12)26/h1,3,5-7,9,12,15-16,25-26H,2,4,8H2,(H,21,22)/t12-,15+,16-/m0/s1
GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333418
PNG
(4-[5-(Cyclobutylmethoxy)-1-methyl-1H-benzimidazol-...)
Show SMILES Cn1cnc2cc(OCC3CCC3)c(cc12)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C19H20ClFN4O2/c20-13-9-11(1-3-14(13)21)5-6-22-18-19-24-10-15(25(19)8-7-23-18)12-2-4-16(26)17(12)27/h1,3,7-10,12,16-17,26-27H,2,4-6H2,(H,22,23)/t12-,16+,17-/m0/s1
GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333420
PNG
(4-[5-(Cyclobutylmethoxy)-1-benzyl-1H-benzimidazol-...)
Show SMILES Cn1cc(-c2cc3n(Cc4ccccc4)cnc3cc2OCC2CCC2)c2cc[nH]c2c1=O
Show InChI InChI=1S/C19H20ClFN4O2/c20-13-3-1-11(9-14(13)21)5-6-22-18-19-24-10-15(25(19)8-7-23-18)12-2-4-16(26)17(12)27/h1,3,7-10,12,16-17,26-27H,2,4-6H2,(H,22,23)/t12-,16+,17-/m0/s1
GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333425
PNG
(4-[5-(Cyclobutylmethoxy)-2-cyclopentyl-1H-benzimid...)
Show SMILES Cn1cc(-c2cc3[nH]c(nc3cc2OCC2CCC2)C2CCCC2)c2cc[nH]c2c1=O
Show InChI InChI=1S/C18H20FN5O2/c19-12-3-1-11(2-4-12)7-8-20-16-18-23-22-17(24(18)10-9-21-16)13-5-6-14(25)15(13)26/h1-4,9-10,13-15,25-26H,5-8H2,(H,20,21)/t13-,14-,15+/m1/s1
GoogleScholar
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PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333416
PNG
(4-[5-(Cyclobutylmethoxy)-1-ethyl-1H-benzimidazol-6...)
Show SMILES CCn1cnc2cc(OCC3CCC3)c(cc12)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C19H21FN4O2/c20-13-3-1-2-12(10-13)6-7-21-18-19-23-11-15(24(19)9-8-22-18)14-4-5-16(25)17(14)26/h1-3,8-11,14,16-17,25-26H,4-7H2,(H,21,22)/t14-,16+,17-/m0/s1
GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333418
PNG
(4-[5-(Cyclobutylmethoxy)-1-methyl-1H-benzimidazol-...)
Show SMILES Cn1cnc2cc(OCC3CCC3)c(cc12)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C19H20ClFN4O2/c20-13-9-11(1-3-14(13)21)5-6-22-18-19-24-10-15(25(19)8-7-23-18)12-2-4-16(26)17(12)27/h1,3,7-10,12,16-17,26-27H,2,4-6H2,(H,22,23)/t12-,16+,17-/m0/s1
GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333420
PNG
(4-[5-(Cyclobutylmethoxy)-1-benzyl-1H-benzimidazol-...)
Show SMILES Cn1cc(-c2cc3n(Cc4ccccc4)cnc3cc2OCC2CCC2)c2cc[nH]c2c1=O
Show InChI InChI=1S/C19H20ClFN4O2/c20-13-3-1-11(9-14(13)21)5-6-22-18-19-24-10-15(25(19)8-7-23-18)12-2-4-16(26)17(12)27/h1,3,7-10,12,16-17,26-27H,2,4-6H2,(H,22,23)/t12-,16+,17-/m0/s1
GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333424
PNG
(4-[5-(Cyclobutylmethoxy)-2-piperidin-1-yl-1H-benzi...)
Show SMILES Cn1cc(-c2cc3[nH]c(nc3cc2OCC2CCC2)N2CCCCC2)c2cc[nH]c2c1=O
Show InChI InChI=1S/C17H17ClFN5O2/c18-10-1-3-12(19)9(7-10)8-21-15-17-23-22-16(24(17)6-5-20-15)11-2-4-13(25)14(11)26/h1,3,5-7,11,13-14,25-26H,2,4,8H2,(H,20,21)/t11-,13-,14+/m1/s1
GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333425
PNG
(4-[5-(Cyclobutylmethoxy)-2-cyclopentyl-1H-benzimid...)
Show SMILES Cn1cc(-c2cc3[nH]c(nc3cc2OCC2CCC2)C2CCCC2)c2cc[nH]c2c1=O
Show InChI InChI=1S/C18H20FN5O2/c19-12-3-1-11(2-4-12)7-8-20-16-18-23-22-17(24(18)10-9-21-16)13-5-6-14(25)15(13)26/h1-4,9-10,13-15,25-26H,5-8H2,(H,20,21)/t13-,14-,15+/m1/s1
GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333408
PNG
(4-[6-(2,4-Difluorophenoxy)-1,2-dimethyl-1H-benzimi...)
Show SMILES Cc1nc2cc(c(Oc3ccc(F)cc3F)cc2n1C)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C17H17ClN4O2S/c18-11-3-1-2-10(6-11)7-20-16-12-8-21-17(22(12)5-4-19-16)15-14(24)13(23)9-25-15/h1-6,8,13-15,23-24H,7,9H2,(H,19,20)/t13-,14-,15-/m1/s1
GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333408
PNG
(4-[6-(2,4-Difluorophenoxy)-1,2-dimethyl-1H-benzimi...)
Show SMILES Cc1nc2cc(c(Oc3ccc(F)cc3F)cc2n1C)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C17H17ClN4O2S/c18-11-3-1-2-10(6-11)7-20-16-12-8-21-17(22(12)5-4-19-16)15-14(24)13(23)9-25-15/h1-6,8,13-15,23-24H,7,9H2,(H,19,20)/t13-,14-,15-/m1/s1
GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333410
PNG
(4-[5-(2,4-Difluorophenoxy)-2-methyl-1H-benzimidazo...)
Show SMILES Cc1nc2cc(Oc3ccc(F)cc3F)c(cc2[nH]1)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C18H18ClN3O2S/c19-12-4-1-3-11(7-12)8-20-13-5-2-6-22-14(9-21-18(13)22)17-16(24)15(23)10-25-17/h1-7,9,15-17,20,23-24H,8,10H2/t15-,16-,17+/m1/s1
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n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333413
PNG
(4-[6-(2,4-Difluorophenoxy)-1H-benzimidazol-5-yl]-6...)
Show SMILES Cn1cc(-c2cc3[nH]cnc3cc2Oc2ccc(F)cc2F)c2cn[nH]c2c1=O
Show InChI InChI=1S/C18H18Cl2N4O2/c19-11-1-3-13(20)10(7-11)8-22-17-18-23-9-14(24(18)6-5-21-17)12-2-4-15(25)16(12)26/h1,3,5-7,9,12,15-16,25-26H,2,4,8H2,(H,21,22)/t12-,15+,16-/m0/s1
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n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333426
PNG
(Ammonium 3-[5-(cyclobutylmethoxy)-6-(6-methyl-7-ox...)
Show SMILES Cn1cc(-c2cc3[nH]c(CCC([O-])=O)nc3cc2OCC2CCC2)c2cc[nH]c2c1=O
Show InChI InChI=1S/C18H20FN5O2/c19-12-3-1-2-11(10-12)6-7-20-16-18-23-22-17(24(18)9-8-21-16)13-4-5-14(25)15(13)26/h1-3,8-10,13-15,25-26H,4-7H2,(H,20,21)/t13-,14-,15+/m1/s1
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n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333406
PNG
(6-(2,4-Difluorophenoxy)-1-methyl-5-(6-methyl-7-oxo...)
Show SMILES Cn1c2cc(Oc3ccc(F)cc3F)c(cc2[nH]c1=O)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C17H16Cl2N4O2S/c18-10-3-1-2-9(4-10)5-20-16-17-21-6-11(23(17)7-13(19)22-16)15-14(25)12(24)8-26-15/h1-4,6-7,12,14-15,24-25H,5,8H2,(H,20,22)/t12-,14-,15+/m1/s1
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n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333407
PNG
(4-[6-(2,4-Difluorophenoxy)-1-methyl-1H-benzimidazo...)
Show SMILES Cn1cnc2cc(c(Oc3ccc(F)cc3F)cc12)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C17H17ClN4O2S/c18-11-4-1-3-10(7-11)8-19-12-5-2-6-22-16(12)20-21-17(22)15-14(24)13(23)9-25-15/h1-7,13-15,19,23-24H,8-9H2/t13-,14-,15-/m1/s1
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n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333407
PNG
(4-[6-(2,4-Difluorophenoxy)-1-methyl-1H-benzimidazo...)
Show SMILES Cn1cnc2cc(c(Oc3ccc(F)cc3F)cc12)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C17H17ClN4O2S/c18-11-4-1-3-10(7-11)8-19-12-5-2-6-22-16(12)20-21-17(22)15-14(24)13(23)9-25-15/h1-7,13-15,19,23-24H,8-9H2/t13-,14-,15-/m1/s1
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Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333422
PNG
(4-[5-(Cyclobutylmethoxy)-1-isopropyl-1H-benzimidaz...)
Show SMILES CC(C)n1cnc2cc(OCC3CCC3)c(cc12)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C17H17Cl2N5O2/c18-10-5-9(6-11(19)7-10)8-21-15-17-23-22-16(24(17)4-3-20-15)12-1-2-13(25)14(12)26/h3-7,12-14,25-26H,1-2,8H2,(H,20,21)/t12-,13-,14+/m1/s1
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n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333410
PNG
(4-[5-(2,4-Difluorophenoxy)-2-methyl-1H-benzimidazo...)
Show SMILES Cc1nc2cc(Oc3ccc(F)cc3F)c(cc2[nH]1)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C18H18ClN3O2S/c19-12-4-1-3-11(7-12)8-20-13-5-2-6-22-14(9-21-18(13)22)17-16(24)15(23)10-25-17/h1-7,9,15-17,20,23-24H,8,10H2/t15-,16-,17+/m1/s1
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n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333411
PNG
(5-(2,4-Difluorophenoxy)-1,3-dimethyl-6-(6-methyl-7...)
Show SMILES Cn1c2cc(Oc3ccc(F)cc3F)c(cc2n(C)c1=O)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C18H19ClN4O2/c19-12-3-1-2-11(8-12)9-21-17-18-22-10-14(23(18)7-6-20-17)13-4-5-15(24)16(13)25/h1-3,6-8,10,13,15-16,24-25H,4-5,9H2,(H,20,21)/t13-,15+,16-/m0/s1
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Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333416
PNG
(4-[5-(Cyclobutylmethoxy)-1-ethyl-1H-benzimidazol-6...)
Show SMILES CCn1cnc2cc(OCC3CCC3)c(cc12)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C19H21FN4O2/c20-13-3-1-2-12(10-13)6-7-21-18-19-23-11-15(24(19)9-8-22-18)14-4-5-16(25)17(14)26/h1-3,8-11,14,16-17,25-26H,4-7H2,(H,21,22)/t14-,16+,17-/m0/s1
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Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333418
PNG
(4-[5-(Cyclobutylmethoxy)-1-methyl-1H-benzimidazol-...)
Show SMILES Cn1cnc2cc(OCC3CCC3)c(cc12)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C19H20ClFN4O2/c20-13-9-11(1-3-14(13)21)5-6-22-18-19-24-10-15(25(19)8-7-23-18)12-2-4-16(26)17(12)27/h1,3,7-10,12,16-17,26-27H,2,4-6H2,(H,22,23)/t12-,16+,17-/m0/s1
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n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333422
PNG
(4-[5-(Cyclobutylmethoxy)-1-isopropyl-1H-benzimidaz...)
Show SMILES CC(C)n1cnc2cc(OCC3CCC3)c(cc12)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C17H17Cl2N5O2/c18-10-5-9(6-11(19)7-10)8-21-15-17-23-22-16(24(17)4-3-20-15)12-1-2-13(25)14(12)26/h3-7,12-14,25-26H,1-2,8H2,(H,20,21)/t12-,13-,14+/m1/s1
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n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333426
PNG
(Ammonium 3-[5-(cyclobutylmethoxy)-6-(6-methyl-7-ox...)
Show SMILES Cn1cc(-c2cc3[nH]c(CCC([O-])=O)nc3cc2OCC2CCC2)c2cc[nH]c2c1=O
Show InChI InChI=1S/C18H20FN5O2/c19-12-3-1-2-11(10-12)6-7-20-16-18-23-22-17(24(18)9-8-21-16)13-4-5-14(25)15(13)26/h1-3,8-10,13-15,25-26H,4-7H2,(H,20,21)/t13-,14-,15+/m1/s1
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n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333405
PNG
(5-(2,4-Difluorophenoxy)-6-(6-methyl-7-oxo-6,7-dihy...)
Show SMILES Cn1cc(-c2cc3[nH]c(=O)[nH]c3cc2Oc2ccc(F)cc2F)c2cc[nH]c2c1=O
Show InChI InChI=1S/C19H19ClN4O2S/c20-11-3-1-2-10(6-11)12-7-13(12)23-18-19-22-8-14(24(19)5-4-21-18)17-16(26)15(25)9-27-17/h1-6,8,12-13,15-17,25-26H,7,9H2,(H,21,23)/t12-,13+,15-,16-,17+/m1/s1
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n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333409
PNG
(4-[5-(2,4-Difluorophenoxy)-1H-benzimidazol-6-yl]-6...)
Show SMILES Cn1cc(-c2cc3[nH]cnc3cc2Oc2ccc(F)cc2F)c2cc[nH]c2c1=O
Show InChI InChI=1S/C18H17Cl2N3O2S/c19-11-3-1-2-10(4-11)6-21-13-5-12(20)8-23-14(7-22-18(13)23)17-16(25)15(24)9-26-17/h1-5,7-8,15-17,21,24-25H,6,9H2/t15-,16-,17+/m1/s1
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Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333412
PNG
(4-(5-(2,4-difluorophenoxy)-1H-benzo[d][1,2,3]triaz...)
Show SMILES Cn1cc(-c2cc3[nH]nnc3cc2Oc2ccc(F)cc2F)c2cc[nH]c2c1=O
Show InChI InChI=1S/C18H18Cl2N4O2/c19-11-5-10(6-12(20)7-11)8-22-17-18-23-9-14(24(18)4-3-21-17)13-1-2-15(25)16(13)26/h3-7,9,13,15-16,25-26H,1-2,8H2,(H,21,22)/t13-,15+,16-/m0/s1
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n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333415
PNG
(4-[5-(Cyclobutylmethoxy)-1H-benzimidazol-6-yl]-6-m...)
Show SMILES Cn1cc(-c2cc3NCNc3cc2OCC2CCC2)c2cc[nH]c2c1=O
Show InChI InChI=1S/C19H21FN4O2/c20-13-3-1-12(2-4-13)7-8-21-18-19-23-11-15(24(19)10-9-22-18)14-5-6-16(25)17(14)26/h1-4,9-11,14,16-17,25-26H,5-8H2,(H,21,22)/t14-,16+,17-/m0/s1
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n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333416
PNG
(4-[5-(Cyclobutylmethoxy)-1-ethyl-1H-benzimidazol-6...)
Show SMILES CCn1cnc2cc(OCC3CCC3)c(cc12)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C19H21FN4O2/c20-13-3-1-2-12(10-13)6-7-21-18-19-23-11-15(24(19)9-8-22-18)14-4-5-16(25)17(14)26/h1-3,8-11,14,16-17,25-26H,4-7H2,(H,21,22)/t14-,16+,17-/m0/s1
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Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333416
PNG
(4-[5-(Cyclobutylmethoxy)-1-ethyl-1H-benzimidazol-6...)
Show SMILES CCn1cnc2cc(OCC3CCC3)c(cc12)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C19H21FN4O2/c20-13-3-1-2-12(10-13)6-7-21-18-19-23-11-15(24(19)9-8-22-18)14-4-5-16(25)17(14)26/h1-3,8-11,14,16-17,25-26H,4-7H2,(H,21,22)/t14-,16+,17-/m0/s1
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n/an/a<100n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333420
PNG
(4-[5-(Cyclobutylmethoxy)-1-benzyl-1H-benzimidazol-...)
Show SMILES Cn1cc(-c2cc3n(Cc4ccccc4)cnc3cc2OCC2CCC2)c2cc[nH]c2c1=O
Show InChI InChI=1S/C19H20ClFN4O2/c20-13-3-1-11(9-14(13)21)5-6-22-18-19-24-10-15(25(19)8-7-23-18)12-2-4-16(26)17(12)27/h1,3,7-10,12,16-17,26-27H,2,4-6H2,(H,22,23)/t12-,16+,17-/m0/s1
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Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)


(Homo sapiens (Human))
BDBM333422
PNG
(4-[5-(Cyclobutylmethoxy)-1-isopropyl-1H-benzimidaz...)
Show SMILES CC(C)n1cnc2cc(OCC3CCC3)c(cc12)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C17H17Cl2N5O2/c18-10-5-9(6-11(19)7-10)8-21-15-17-23-22-16(24(17)4-3-20-15)12-1-2-13(25)14(12)26/h3-7,12-14,25-26H,1-2,8H2,(H,20,21)/t12-,13-,14+/m1/s1
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Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333420
PNG
(4-[5-(Cyclobutylmethoxy)-1-benzyl-1H-benzimidazol-...)
Show SMILES Cn1cc(-c2cc3n(Cc4ccccc4)cnc3cc2OCC2CCC2)c2cc[nH]c2c1=O
Show InChI InChI=1S/C19H20ClFN4O2/c20-13-3-1-11(9-14(13)21)5-6-22-18-19-24-10-15(25(19)8-7-23-18)12-2-4-16(26)17(12)27/h1,3,7-10,12,16-17,26-27H,2,4-6H2,(H,22,23)/t12-,16+,17-/m0/s1
GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a 550n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)


(Homo sapiens (Human))
BDBM333411
PNG
(5-(2,4-Difluorophenoxy)-1,3-dimethyl-6-(6-methyl-7...)
Show SMILES Cn1c2cc(Oc3ccc(F)cc3F)c(cc2n(C)c1=O)-c1cn(C)c(=O)c2[nH]ccc12
Show InChI InChI=1S/C18H19ClN4O2/c19-12-3-1-2-11(8-12)9-21-17-18-22-10-14(23(18)7-6-20-17)13-4-5-15(24)16(13)25/h1-3,6-8,10,13,15-16,24-25H,4-5,9H2,(H,20,21)/t13-,15+,16-/m0/s1
GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a 550n/an/an/an/an/an/a



Incyte Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9737516 (2017)

More data for this
Ligand-Target Pair
* indicates data uncertainty>20%