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Patent code US9745317

Compile Data Set for Download or QSAR
Found 28 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337378
PNG
(5-{4-[(3-Hydroxy-2,3-dihydrofuro[3,2-c]pyridin-4-y...)
Show SMILES Cc1cc(Oc2nccc3OCC(O)c23)ccc1-c1c(C)n[nH]c(=O)c1C
Show InChI InChI=1S/C20H19N3O4/c1-10-8-13(27-20-18-15(24)9-26-16(18)6-7-21-20)4-5-14(10)17-11(2)19(25)23-22-12(17)3/h4-8,15,24H,9H2,1-3H3,(H,23,25)
KEGG

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US Patent
4.80n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337370
PNG
(5-[4-(2,3-dihydro-1H-pyrrolo[3,2-c]pyridin-4-yloxy...)
Show SMILES Cc1cc(Oc2nccc3NCCc23)ccc1-c1c(C)n[nH]c(=O)c1C
Show InChI InChI=1S/C20H20N4O2/c1-11-10-14(26-20-16-6-8-21-17(16)7-9-22-20)4-5-15(11)18-12(2)19(25)24-23-13(18)3/h4-5,7,9-10,21H,6,8H2,1-3H3,(H,24,25)
KEGG

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8.40n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337374
PNG
(6-[4-(2,3-Dihydro-1H-pyrrolo[3,2-c]pyridin-4-yloxy...)
Show SMILES CC(C)c1cc(C(C)C)c(c(c1)C(C)C)-c1c(C)c(C)c(C)c(C)c1P(C(C)(C)C)C(C)(C)C
Show InChI InChI=1S/C33H53P/c1-19(2)26-17-27(20(3)4)30(28(18-26)21(5)6)29-24(9)22(7)23(8)25(10)31(29)34(32(11,12)13)33(14,15)16/h17-21H,1-16H3
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11.1n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337368
PNG
((+)-5-[4-(2,3-dihydrofuro[3,2-c]pyridin-4-yloxy)-2...)
Show SMILES Cc1cc(Oc2nccc3OCCc23)ccc1-c1c(C)n[nH]c(=O)c1C
Show InChI InChI=1S/C20H19N3O3/c1-11-10-14(26-20-16-7-9-25-17(16)6-8-21-20)4-5-15(11)18-12(2)19(24)23-22-13(18)3/h4-6,8,10H,7,9H2,1-3H3,(H,23,24)
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12.6n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337369
PNG
((−)-5-[4-(2,3-dihydrofuro[3,2-c]pyridin-4-yl...)
Show SMILES Cc1cc(Oc2nccc3OCCc23)ccc1-c1c(C)n[nH]c(=O)c1C
Show InChI InChI=1S/C20H19N3O3/c1-11-10-14(26-20-16-7-9-25-17(16)6-8-21-20)4-5-15(11)18-12(2)19(24)23-22-13(18)3/h4-6,8,10H,7,9H2,1-3H3,(H,23,24)
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12.7n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337367
PNG
(5-[4-(2,3-dihydrofuro[3,2-c]pyridin-4-yloxy)-2- me...)
Show SMILES Cc1cc(Oc2nccc3OCCc23)ccc1-c1c(C)n[nH]c(=O)c1C
Show InChI InChI=1S/C20H19N3O3/c1-11-10-14(26-20-16-7-9-25-17(16)6-8-21-20)4-5-15(11)18-12(2)19(24)23-22-13(18)3/h4-6,8,10H,7,9H2,1-3H3,(H,23,24)
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14n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337366
PNG
(5-[4-(2,3-Dihydro-1H-pyrrolo[3,2-c]pyridin-4-yloxy...)
Show SMILES Cc1nn(C2CCCCO2)c(=O)c(C)c1-c1ccc(Oc2nccc3N(CCc23)C(c2ccccc2)(c2ccccc2)c2ccccc2)cc1
Show InChI InChI=1S/C43H40N4O3/c1-30-40(31(2)45-47(42(30)48)39-20-12-13-29-49-39)32-21-23-36(24-22-32)50-41-37-26-28-46(38(37)25-27-44-41)43(33-14-6-3-7-15-33,34-16-8-4-9-17-34)35-18-10-5-11-19-35/h3-11,14-19,21-25,27,39H,12-13,20,26,28-29H2,1-2H3
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14n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337377
PNG
(4,6-Dimethyl-5-[2-methyl-4-(1,2,3,4-tetrahydro-1,6...)
Show SMILES Cc1cc(Oc2nccc3N(Cc4ccccc4)CCCc23)ccc1-c1c(C)nn(C2CCCCO2)c(=O)c1C
Show InChI InChI=1S/C33H36N4O3/c1-22-20-26(14-15-27(22)31-23(2)33(38)37(35-24(31)3)30-13-7-8-19-39-30)40-32-28-12-9-18-36(29(28)16-17-34-32)21-25-10-5-4-6-11-25/h4-6,10-11,14-17,20,30H,7-9,12-13,18-19,21H2,1-3H3
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18.1n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337379
PNG
(4-[4-(4,6-Dimethylpyrimidin-5-yl)-3-methylphenoxy]...)
Show SMILES CC(C)c1cc(C(C)C)c(c(c1)C(C)C)-c1c(C)c(C)c(C)c(C)c1P(C(C)(C)C)C(C)(C)C
Show InChI InChI=1S/C33H53P/c1-19(2)26-17-27(20(3)4)30(28(18-26)21(5)6)29-24(9)22(7)23(8)25(10)31(29)34(32(11,12)13)33(14,15)16/h17-21H,1-16H3
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28.9n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337370
PNG
(5-[4-(2,3-dihydro-1H-pyrrolo[3,2-c]pyridin-4-yloxy...)
Show SMILES Cc1cc(Oc2nccc3NCCc23)ccc1-c1c(C)n[nH]c(=O)c1C
Show InChI InChI=1S/C20H20N4O2/c1-11-10-14(26-20-16-6-8-21-17(16)7-9-22-20)4-5-15(11)18-12(2)19(25)24-23-13(18)3/h4-5,7,9-10,21H,6,8H2,1-3H3,(H,24,25)
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35.6n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337389
PNG
(US9745317, 27)
Show SMILES Cc1c(-c2ccc(Oc3ncnc4NCCc34)cc2)n(C)c(=O)[nH]c1=O
Show InChI InChI=1S/C18H17N5O3/c1-10-14(23(2)18(25)22-16(10)24)11-3-5-12(6-4-11)26-17-13-7-8-19-15(13)20-9-21-17/h3-6,9H,7-8H2,1-2H3,(H,19,20,21)(H,22,24,25)
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44.4n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337375
PNG
(6-[4-(2,3-Dihydrofuro[3,2-c]pyridin-4-yloxy)phenyl...)
Show SMILES CC(C)c1cc(C(C)C)c(c(c1)C(C)C)-c1c(C)c(C)c(C)c(C)c1P(C(C)(C)C)C(C)(C)C
Show InChI InChI=1S/C33H53P/c1-19(2)26-17-27(20(3)4)30(28(18-26)21(5)6)29-24(9)22(7)23(8)25(10)31(29)34(32(11,12)13)33(14,15)16/h17-21H,1-16H3
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46.1n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337370
PNG
(5-[4-(2,3-dihydro-1H-pyrrolo[3,2-c]pyridin-4-yloxy...)
Show SMILES Cc1cc(Oc2nccc3NCCc23)ccc1-c1c(C)n[nH]c(=O)c1C
Show InChI InChI=1S/C20H20N4O2/c1-11-10-14(26-20-16-6-8-21-17(16)7-9-22-20)4-5-15(11)18-12(2)19(25)24-23-13(18)3/h4-5,7,9-10,21H,6,8H2,1-3H3,(H,24,25)
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50.5n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337365
PNG
(5-[4-(2,3-Dihydrofuro[3,2-c]pyridin-4-yloxy)phenyl...)
Show SMILES CC1(C)c2cccc(P(c3ccccc3)c3ccccc3)c2Oc2c(cccc12)P(c1ccccc1)c1ccccc1
Show InChI InChI=1S/C39H32OP2/c1-39(2)33-25-15-27-35(41(29-17-7-3-8-18-29)30-19-9-4-10-20-30)37(33)40-38-34(39)26-16-28-36(38)42(31-21-11-5-12-22-31)32-23-13-6-14-24-32/h3-28H,1-2H3
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52n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337380
PNG
(US9745317, 18)
Show SMILES Cc1cc(Oc2nccc3OCCc23)ccc1-c1c(C)ncc2nccn12
Show InChI InChI=1S/C21H18N4O2/c1-13-11-15(27-21-17-6-10-26-18(17)5-7-23-21)3-4-16(13)20-14(2)24-12-19-22-8-9-25(19)20/h3-5,7-9,11-12H,6,10H2,1-2H3
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52.1n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337373
PNG
(5-[4-(6, 7-Dihydro-5H-pyrrolo[2, 3-d]pyrimidin-4-y...)
Show SMILES COc1ccc(CN2CCc3c2ncnc3Oc2ccc(cc2)-c2c(C)nn(C3CCCCO3)c(=O)c2C)cc1
Show InChI InChI=1S/C31H33N5O4/c1-20-28(21(2)34-36(31(20)37)27-6-4-5-17-39-27)23-9-13-25(14-10-23)40-30-26-15-16-35(29(26)32-19-33-30)18-22-7-11-24(38-3)12-8-22/h7-14,19,27H,4-6,15-18H2,1-3H3
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60.4n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337376
PNG
(5-[4-(3,4-Dihydro-2H-pyrano[3,2-c]pyridin-5-yloxy)...)
Show SMILES CC1(C)c2cccc(P(c3ccccc3)c3ccccc3)c2Cc2c(cccc12)P(c1ccccc1)c1ccccc1
Show InChI InChI=1S/C40H34P2/c1-40(2)36-25-15-27-38(41(30-17-7-3-8-18-30)31-19-9-4-10-20-31)34(36)29-35-37(40)26-16-28-39(35)42(32-21-11-5-12-22-32)33-23-13-6-14-24-33/h3-28H,29H2,1-2H3
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70.3n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337386
PNG
(US9745317, 24 | US9745317, 25)
Show SMILES Cc1cc(Oc2nccc3NCCc23)ccc1-c1c(C)ncc(=O)n1C
Show InChI InChI=1S/C20H20N4O2/c1-12-10-14(26-20-16-6-8-21-17(16)7-9-22-20)4-5-15(12)19-13(2)23-11-18(25)24(19)3/h4-5,7,9-11,21H,6,8H2,1-3H3
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75.8n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337363
PNG
(4-[4-(4,6-Dimethylpyrimidin-5-yl)-3-methylphenoxy]...)
Show SMILES Cc1cc(Oc2nccc3OCCc23)ccc1-c1c(C)ncnc1C
Show InChI InChI=1S/C20H19N3O2/c1-12-10-15(25-20-17-7-9-24-18(17)6-8-21-20)4-5-16(12)19-13(2)22-11-23-14(19)3/h4-6,8,10-11H,7,9H2,1-3H3
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76.8n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337364
PNG
(4-[4-(4,6-Dimethylpyrimidin-5-yl)-3-methylphenoxy]...)
Show SMILES CC1=C(C(C)=[N](C)C=N1)c1ccc(Oc2nccc3N(CCc23)C2CCCCO2)cc1C
Show InChI InChI=1S/C26H31N4O2/c1-17-15-20(8-9-21(17)25-18(2)28-16-29(4)19(25)3)32-26-22-11-13-30(23(22)10-12-27-26)24-7-5-6-14-31-24/h8-10,12,15-16,24H,5-7,11,13-14H2,1-4H3
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78.1n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337383
PNG
(US9745317, 21 | US9745317, 22 | US9745317, 23)
Show SMILES Cc1cc(Oc2nccc3OCCc23)ccc1-c1c(C)ncc(=O)n1C
Show InChI InChI=1S/C20H19N3O3/c1-12-10-14(26-20-16-7-9-25-17(16)6-8-21-20)4-5-15(12)19-13(2)22-11-18(24)23(19)3/h4-6,8,10-11H,7,9H2,1-3H3
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82.5n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337381
PNG
(US9745317, 19)
Show SMILES Cc1cc(Oc2ncnc3NCCc23)ccc1-c1c(C)ncnc1C
Show InChI InChI=1S/C19H19N5O/c1-11-8-14(25-19-16-6-7-20-18(16)23-10-24-19)4-5-15(11)17-12(2)21-9-22-13(17)3/h4-5,8-10H,6-7H2,1-3H3,(H,20,23,24)
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156n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337388
PNG
(US9745317, 26)
Show SMILES Cc1n[nH]c(=O)c(C)c1-c1ccc(Oc2nccc3OCCc23)cc1C#N
Show InChI InChI=1S/C20H16N4O3/c1-11-18(12(2)23-24-19(11)25)15-4-3-14(9-13(15)10-21)27-20-16-6-8-26-17(16)5-7-22-20/h3-5,7,9H,6,8H2,1-2H3,(H,24,25)
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UniProtKB/SwissProt

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US Patent
162n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337386
PNG
(US9745317, 24 | US9745317, 25)
Show SMILES Cc1cc(Oc2nccc3NCCc23)ccc1-c1c(C)ncc(=O)n1C
Show InChI InChI=1S/C20H20N4O2/c1-12-10-14(26-20-16-6-8-21-17(16)7-9-22-20)4-5-15(12)19-13(2)23-11-18(25)24(19)3/h4-5,7,9-11,21H,6,8H2,1-3H3
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201n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337383
PNG
(US9745317, 21 | US9745317, 22 | US9745317, 23)
Show SMILES Cc1cc(Oc2nccc3OCCc23)ccc1-c1c(C)ncc(=O)n1C
Show InChI InChI=1S/C20H19N3O3/c1-12-10-14(26-20-16-7-9-25-17(16)6-8-21-20)4-5-15(12)19-13(2)22-11-18(24)23(19)3/h4-6,8,10-11H,7,9H2,1-3H3
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202n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337390
PNG
(US9745317, 28)
Show SMILES Cc1c(-c2ccc(Oc3ncnc4CCCc34)cc2)n(C)c(=O)[nH]c1=O
Show InChI InChI=1S/C19H18N4O3/c1-11-16(23(2)19(25)22-17(11)24)12-6-8-13(9-7-12)26-18-14-4-3-5-15(14)20-10-21-18/h6-10H,3-5H2,1-2H3,(H,22,24,25)
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202n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337382
PNG
(US9745317, 20)
Show SMILES Cc1cc(Oc2ncnc3CCCc23)ccc1-c1c(C)ncnc1C
Show InChI InChI=1S/C20H20N4O/c1-12-9-15(25-20-17-5-4-6-18(17)23-11-24-20)7-8-16(12)19-13(2)21-10-22-14(19)3/h7-11H,4-6H2,1-3H3
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446n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
Dopamine D1 receptor


(Homo sapiens (Human))
BDBM337383
PNG
(US9745317, 21 | US9745317, 22 | US9745317, 23)
Show SMILES Cc1cc(Oc2nccc3OCCc23)ccc1-c1c(C)ncc(=O)n1C
Show InChI InChI=1S/C20H19N3O3/c1-12-10-14(26-20-16-7-9-25-17(16)6-8-21-20)4-5-15(12)19-13(2)22-11-18(24)23(19)3/h4-6,8,10-11H,7,9H2,1-3H3
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706n/an/an/an/an/an/an/an/a



Pfizer Inc.

US Patent


Assay Description
D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...


US Patent US9745317 (2017)

More data for this
Ligand-Target Pair
* indicates data uncertainty>20%