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Patent code US9796664

Compile Data Set for Download or QSAR
Found 27 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Histone deacetylase 3


(Homo sapiens (Human))
BDBM207629
PNG
(US9265734, R01 | US9796664, Compound R01)
Show SMILES Cc1ccc(cc1)C(=O)NCCCCCC(=O)Nc1ccccc1N
Show InChI InChI=1S/C20H25N3O2/c1-15-10-12-16(13-11-15)20(25)22-14-6-2-3-9-19(24)23-18-8-5-4-7-17(18)21/h4-5,7-8,10-13H,2-3,6,9,14,21H2,1H3,(H,22,25)(H,23,24)
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n/an/a 300n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))
BDBM19410
PNG
(CHEMBL27759 | MS-275 | US9265734, MS-275 | US97966...)
Show SMILES Nc1ccccc1NC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1
Show InChI InChI=1S/C21H20N4O3/c22-18-5-1-2-6-19(18)25-20(26)17-9-7-15(8-10-17)13-24-21(27)28-14-16-4-3-11-23-12-16/h1-12H,13-14,22H2,(H,24,27)(H,25,26)
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n/an/a 590n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))
BDBM207628
PNG
(US9265734, RGFA8 | US9796664, Compound RGFA8)
Show SMILES Cc1ccc(NC(=O)CCCCCC(=O)Nc2ccccc2N)cc1
Show InChI InChI=1S/C20H25N3O2/c1-15-11-13-16(14-12-15)22-19(24)9-3-2-4-10-20(25)23-18-8-6-5-7-17(18)21/h5-8,11-14H,2-4,9-10,21H2,1H3,(H,22,24)(H,23,25)
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n/an/a 700n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))
BDBM207628
PNG
(US9265734, RGFA8 | US9796664, Compound RGFA8)
Show SMILES Cc1ccc(NC(=O)CCCCCC(=O)Nc2ccccc2N)cc1
Show InChI InChI=1S/C20H25N3O2/c1-15-11-13-16(14-12-15)22-19(24)9-3-2-4-10-20(25)23-18-8-6-5-7-17(18)21/h5-8,11-14H,2-4,9-10,21H2,1H3,(H,22,24)(H,23,25)
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n/an/a 700n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 2


(Homo sapiens (Human))
BDBM19410
PNG
(CHEMBL27759 | MS-275 | US9265734, MS-275 | US97966...)
Show SMILES Nc1ccccc1NC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1
Show InChI InChI=1S/C21H20N4O3/c22-18-5-1-2-6-19(18)25-20(26)17-9-7-15(8-10-17)13-24-21(27)28-14-16-4-3-11-23-12-16/h1-12H,13-14,22H2,(H,24,27)(H,25,26)
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n/an/a 720n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))
BDBM207632
PNG
(US9265734, R03 | US9796664, Compound R03)
Show SMILES Cc1ccc(cc1)C(=O)NCCCCCC(=O)Nc1ccc(F)cc1N
Show InChI InChI=1S/C20H24FN3O2/c1-14-6-8-15(9-7-14)20(26)23-12-4-2-3-5-19(25)24-18-11-10-16(21)13-17(18)22/h6-11,13H,2-5,12,22H2,1H3,(H,23,26)(H,24,25)
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n/an/a 800n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))
BDBM207634
PNG
(US9265734, R05 | US9796664, Compound R05)
Show SMILES Cc1ccc(cc1)C(=O)Nc1cccc(\C=C\C(=O)Nc2ccc(F)cc2N)c1
Show InChI InChI=1S/C23H20FN3O2/c1-15-5-8-17(9-6-15)23(29)26-19-4-2-3-16(13-19)7-12-22(28)27-21-11-10-18(24)14-20(21)25/h2-14H,25H2,1H3,(H,26,29)(H,27,28)/b12-7+
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n/an/a 1.40E+3n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))
BDBM207636
PNG
(US9265734, R07 | US9796664, Compound R07)
Show SMILES Nc1cc(F)ccc1NC(=O)CCCCCNC(=O)c1ccc(F)cc1
Show InChI InChI=1S/C19H21F2N3O2/c20-14-7-5-13(6-8-14)19(26)23-11-3-1-2-4-18(25)24-17-10-9-15(21)12-16(17)22/h5-10,12H,1-4,11,22H2,(H,23,26)(H,24,25)
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n/an/a 1.60E+3n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))
BDBM207635
PNG
(US9265734, R06 | US9796664, Compound R06)
Show SMILES Nc1ccc(F)cc1NC(=O)CCCCCNC(=O)c1ccc(F)cc1
Show InChI InChI=1S/C19H21F2N3O2/c20-14-7-5-13(6-8-14)19(26)23-11-3-1-2-4-18(25)24-17-12-15(21)9-10-16(17)22/h5-10,12H,1-4,11,22H2,(H,23,26)(H,24,25)
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n/an/a 1.80E+3n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 2


(Homo sapiens (Human))
BDBM207629
PNG
(US9265734, R01 | US9796664, Compound R01)
Show SMILES Cc1ccc(cc1)C(=O)NCCCCCC(=O)Nc1ccccc1N
Show InChI InChI=1S/C20H25N3O2/c1-15-10-12-16(13-11-15)20(25)22-14-6-2-3-9-19(24)23-18-8-5-4-7-17(18)21/h4-5,7-8,10-13H,2-3,6,9,14,21H2,1H3,(H,22,25)(H,23,24)
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n/an/a 1.98E+3n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))
BDBM207628
PNG
(US9265734, RGFA8 | US9796664, Compound RGFA8)
Show SMILES Cc1ccc(NC(=O)CCCCCC(=O)Nc2ccccc2N)cc1
Show InChI InChI=1S/C20H25N3O2/c1-15-11-13-16(14-12-15)22-19(24)9-3-2-4-10-20(25)23-18-8-6-5-7-17(18)21/h5-8,11-14H,2-4,9-10,21H2,1H3,(H,22,24)(H,23,25)
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n/an/a 2.00E+3n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))
BDBM207628
PNG
(US9265734, RGFA8 | US9796664, Compound RGFA8)
Show SMILES Cc1ccc(NC(=O)CCCCCC(=O)Nc2ccccc2N)cc1
Show InChI InChI=1S/C20H25N3O2/c1-15-11-13-16(14-12-15)22-19(24)9-3-2-4-10-20(25)23-18-8-6-5-7-17(18)21/h5-8,11-14H,2-4,9-10,21H2,1H3,(H,22,24)(H,23,25)
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n/an/a 2.00E+3n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))
BDBM207631
PNG
(US9265734, R02 | US9796664, Compound R02)
Show SMILES Nc1cc(F)ccc1NC(=O)CCCCCNC(=O)c1nccs1
Show InChI InChI=1S/C16H19FN4O2S/c17-11-5-6-13(12(18)10-11)21-14(22)4-2-1-3-7-19-15(23)16-20-8-9-24-16/h5-6,8-10H,1-4,7,18H2,(H,19,23)(H,21,22)
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n/an/a 2.30E+3n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))
BDBM207629
PNG
(US9265734, R01 | US9796664, Compound R01)
Show SMILES Cc1ccc(cc1)C(=O)NCCCCCC(=O)Nc1ccccc1N
Show InChI InChI=1S/C20H25N3O2/c1-15-10-12-16(13-11-15)20(25)22-14-6-2-3-9-19(24)23-18-8-5-4-7-17(18)21/h4-5,7-8,10-13H,2-3,6,9,14,21H2,1H3,(H,22,25)(H,23,24)
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n/an/a 2.40E+3n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))
BDBM19410
PNG
(CHEMBL27759 | MS-275 | US9265734, MS-275 | US97966...)
Show SMILES Nc1ccccc1NC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1
Show InChI InChI=1S/C21H20N4O3/c22-18-5-1-2-6-19(18)25-20(26)17-9-7-15(8-10-17)13-24-21(27)28-14-16-4-3-11-23-12-16/h1-12H,13-14,22H2,(H,24,27)(H,25,26)
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n/an/a 3.20E+3n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))
BDBM207637
PNG
(BDBM207672 | US9265734, R08 | US9796664, Compound ...)
Show SMILES Nc1ccccc1NC(=O)CCCCCNS(=O)(=O)c1ccc(F)cc1
Show InChI InChI=1S/C18H22FN3O3S/c19-14-9-11-15(12-10-14)26(24,25)21-13-5-1-2-8-18(23)22-17-7-4-3-6-16(17)20/h3-4,6-7,9-12,21H,1-2,5,8,13,20H2,(H,22,23)
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n/an/a 3.60E+3n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 2


(Homo sapiens (Human))
BDBM207628
PNG
(US9265734, RGFA8 | US9796664, Compound RGFA8)
Show SMILES Cc1ccc(NC(=O)CCCCCC(=O)Nc2ccccc2N)cc1
Show InChI InChI=1S/C20H25N3O2/c1-15-11-13-16(14-12-15)22-19(24)9-3-2-4-10-20(25)23-18-8-6-5-7-17(18)21/h5-8,11-14H,2-4,9-10,21H2,1H3,(H,22,24)(H,23,25)
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n/an/a 3.73E+3n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))
BDBM207635
PNG
(US9265734, R06 | US9796664, Compound R06)
Show SMILES Nc1ccc(F)cc1NC(=O)CCCCCNC(=O)c1ccc(F)cc1
Show InChI InChI=1S/C19H21F2N3O2/c20-14-7-5-13(6-8-14)19(26)23-11-3-1-2-4-18(25)24-17-12-15(21)9-10-16(17)22/h5-10,12H,1-4,11,22H2,(H,23,26)(H,24,25)
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n/an/a 5.70E+3n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))
BDBM207638
PNG
(BDBM207673 | US9265734, R09 | US9796664, Compound ...)
Show SMILES Nc1cc(F)ccc1NC(=O)CCCCCNS(=O)(=O)c1ccc(F)cc1
Show InChI InChI=1S/C18H21F2N3O3S/c19-13-5-8-15(9-6-13)27(25,26)22-11-3-1-2-4-18(24)23-17-10-7-14(20)12-16(17)21/h5-10,12,22H,1-4,11,21H2,(H,23,24)
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n/an/a 7.30E+3n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))
BDBM207632
PNG
(US9265734, R03 | US9796664, Compound R03)
Show SMILES Cc1ccc(cc1)C(=O)NCCCCCC(=O)Nc1ccc(F)cc1N
Show InChI InChI=1S/C20H24FN3O2/c1-14-6-8-15(9-7-14)20(26)23-12-4-2-3-5-19(25)24-18-11-10-16(21)13-17(18)22/h6-11,13H,2-5,12,22H2,1H3,(H,23,26)(H,24,25)
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n/an/a 8.20E+3n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))
BDBM207633
PNG
(US9265734, R04 | US9796664, Compound R04)
Show SMILES Nc1cc(F)ccc1NC(=O)CCCCCNC(=O)CN1CCOCC1
Show InChI InChI=1S/C18H27FN4O3/c19-14-5-6-16(15(20)12-14)22-17(24)4-2-1-3-7-21-18(25)13-23-8-10-26-11-9-23/h5-6,12H,1-4,7-11,13,20H2,(H,21,25)(H,22,24)
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n/an/a 1.40E+4n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))
BDBM207636
PNG
(US9265734, R07 | US9796664, Compound R07)
Show SMILES Nc1cc(F)ccc1NC(=O)CCCCCNC(=O)c1ccc(F)cc1
Show InChI InChI=1S/C19H21F2N3O2/c20-14-7-5-13(6-8-14)19(26)23-11-3-1-2-4-18(25)24-17-10-9-15(21)12-16(17)22/h5-10,12H,1-4,11,22H2,(H,23,26)(H,24,25)
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n/an/a 1.80E+4n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))
BDBM207631
PNG
(US9265734, R02 | US9796664, Compound R02)
Show SMILES Nc1cc(F)ccc1NC(=O)CCCCCNC(=O)c1nccs1
Show InChI InChI=1S/C16H19FN4O2S/c17-11-5-6-13(12(18)10-11)21-14(22)4-2-1-3-7-19-15(23)16-20-8-9-24-16/h5-6,8-10H,1-4,7,18H2,(H,19,23)(H,21,22)
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n/an/a 1.80E+4n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))
BDBM207637
PNG
(BDBM207672 | US9265734, R08 | US9796664, Compound ...)
Show SMILES Nc1ccccc1NC(=O)CCCCCNS(=O)(=O)c1ccc(F)cc1
Show InChI InChI=1S/C18H22FN3O3S/c19-14-9-11-15(12-10-14)26(24,25)21-13-5-1-2-8-18(23)22-17-7-4-3-6-16(17)20/h3-4,6-7,9-12,21H,1-2,5,8,13,20H2,(H,22,23)
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n/an/a 2.40E+4n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))
BDBM207633
PNG
(US9265734, R04 | US9796664, Compound R04)
Show SMILES Nc1cc(F)ccc1NC(=O)CCCCCNC(=O)CN1CCOCC1
Show InChI InChI=1S/C18H27FN4O3/c19-14-5-6-16(15(20)12-14)22-17(24)4-2-1-3-7-21-18(25)13-23-8-10-26-11-9-23/h5-6,12H,1-4,7-11,13,20H2,(H,21,25)(H,22,24)
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n/an/a>3.00E+4n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))
BDBM207638
PNG
(BDBM207673 | US9265734, R09 | US9796664, Compound ...)
Show SMILES Nc1cc(F)ccc1NC(=O)CCCCCNS(=O)(=O)c1ccc(F)cc1
Show InChI InChI=1S/C18H21F2N3O3S/c19-13-5-8-15(9-6-13)27(25,26)22-11-3-1-2-4-18(24)23-17-10-7-14(20)12-16(17)21/h5-10,12,22H,1-4,11,21H2,(H,23,24)
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n/an/a>3.00E+4n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))
BDBM207634
PNG
(US9265734, R05 | US9796664, Compound R05)
Show SMILES Cc1ccc(cc1)C(=O)Nc1cccc(\C=C\C(=O)Nc2ccc(F)cc2N)c1
Show InChI InChI=1S/C23H20FN3O2/c1-15-5-8-17(9-6-15)23(29)26-19-4-2-3-16(13-19)7-12-22(28)27-21-11-10-18(24)14-20(21)25/h2-14H,25H2,1H3,(H,26,29)(H,27,28)/b12-7+
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n/an/a 3.00E+4n/an/an/an/an/an/a



BIOMARIN PHARMACEUTICAL INC.

US Patent


Assay Description
HDAC inhibition assays can be performed, e.g., in a cell, in a cell extract, or in a cell-free mixture. Exemplary HDAC inhibition assays are describe...


US Patent US9796664 (2017)

More data for this
Ligand-Target Pair
* indicates data uncertainty>20%