Compile Data Set for Download or QSAR
maximum 50k data
Found 36 Enz. Inhib. hit(s) with all data for entry = 2048
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101734(US9695160, 31 | US9796707, Compound 31)
Affinity DataIC50:  1.90nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101825(US9695160, 39 | US9796707, Compound 39)
Affinity DataIC50:  2.60nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM221074(SPHINX31 | US9695160, 12 | US9796707, Compound 12)
Affinity DataIC50:  3.18nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101676(US9695160, 20 | US9796707, Compound 20)
Affinity DataIC50:  4.40nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101690(US9695160, 21 | US9796707, Compound 21)
Affinity DataIC50:  4.60nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101824(US9695160, 38 | US9796707, Compound 38)
Affinity DataIC50:  5nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101654(US9695160, 14 | US9796707, Compound 14)
Affinity DataIC50:  7.18nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101713(US9695160, 25 | US9796707, Compound 25)
Affinity DataIC50:  13.5nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101671(US9695160, 18 | US9796707, Compound 18)
Affinity DataIC50:  13.9nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101674(US9695160, 19 | US9796707, Compound 19)
Affinity DataIC50:  14.1nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101695(US9695160, 22 | US9796707, Compound 22)
Affinity DataIC50:  14.8nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101657(US9695160, 15 | US9796707, Compound 15)
Affinity DataIC50:  16.6nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101649(US9695160, 13 | US9796707, Compound 13)
Affinity DataIC50:  17.2nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101659(US9695160, 16 | US9796707, Compound 16)
Affinity DataIC50:  38.2nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM221073(SPHINX scaffold, 3 | US9695160, SPHINX7 | US979670...)
Affinity DataIC50:  54.7nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101660(US9695160, 17 | US9796707, Compound 17)
Affinity DataIC50:  111nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101832(US9695160, 45 | US9796707, Compound 45)
Affinity DataIC50:  119nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101829(US10696661, Compound 74 | US9695160, 42 | US979670...)
Affinity DataIC50:  164nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101815(US9695160, 36 | US9796707, Compound 36)
Affinity DataIC50:  170nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101830(US9695160, 43 | US9796707, Compound 43)
Affinity DataIC50:  183nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101822(US9695160, 37 | US9796707, Compound 37)
Affinity DataIC50:  323nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101728(US9695160, 30 | US9796707, Compound 30)
Affinity DataIC50:  336nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM221070(SPHINX | US9695160, SPHINX | US9796707, Reference ...)
Affinity DataIC50:  440nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101828(US9695160, 41 | US9796707, Compound 41)
Affinity DataIC50:  493nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101737(US9695160, 32 | US9796707, Compound 32)
Affinity DataIC50:  1.55E+3nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101703(US9695160, 24 | US9796707, Compound 24)
Affinity DataIC50:  3.51E+3nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101696(US9695160, 23 | US9796707, Compound 23)
Affinity DataIC50:  4.01E+3nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101739(US9695160, 33 | US9796707, Compound 33)
Affinity DataIC50:  4.03E+3nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101826(US9695160, 40 | US9796707, Compound 40)
Affinity DataIC50:  4.69E+3nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101740(US9695160, 34 | US9796707, Compound 34)
Affinity DataIC50:  5.31E+3nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101831(US9695160, 44 | US9796707, Compound 44)
Affinity DataIC50:  8.41E+3nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101722(US9695160, 29 | US9796707, Compound 29)
Affinity DataIC50:  1.00E+4nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101720(US9695160, 28 | US9796707, Compound 28)
Affinity DataIC50:  1.00E+4nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101715(US9695160, 27 | US9796707, Compound 27)
Affinity DataIC50:  1.00E+4nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101714(US9695160, 26 | US9796707, Compound 26)
Affinity DataIC50:  1.00E+4nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM351702(US9796707, Compound 35)
Affinity DataIC50:  1.00E+4nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent