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Patent code US9850257

Compile Data Set for Download or QSAR
Found 26 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363505
PNG
(9-(3,5-Dimethylisoxazol-4-yl)-6-methoxy-3-pyridin-...)
Show SMILES COc1nn2C(COc3c(ccc1c23)-c1c(C)noc1C)c1cccnc1
Show InChI InChI=1/C20H18N4O3/c1-11-17(12(2)27-23-11)14-6-7-15-18-19(14)26-10-16(13-5-4-8-21-9-13)24(18)22-20(15)25-3/h4-9,16H,10H2,1-3H3
PDB

GoogleScholar
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PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363499
PNG
(9-(3,5-Dimethylisoxazol-4-yl)-5-methyl-3-pyridin-2...)
Show SMILES Cc1noc(C)c1-c1ccc2c3c1OCC(c1ccccn1)n3n(C)c2=O
Show InChI InChI=1/C20H18N4O3/c1-11-17(12(2)27-22-11)13-7-8-14-18-19(13)26-10-16(15-6-4-5-9-21-15)24(18)23(3)20(14)25/h4-9,16H,10H2,1-3H3
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363505
PNG
(9-(3,5-Dimethylisoxazol-4-yl)-6-methoxy-3-pyridin-...)
Show SMILES COc1nn2C(COc3c(ccc1c23)-c1c(C)noc1C)c1cccnc1
Show InChI InChI=1/C20H18N4O3/c1-11-17(12(2)27-23-11)14-6-7-15-18-19(14)26-10-16(13-5-4-8-21-9-13)24(18)22-20(15)25-3/h4-9,16H,10H2,1-3H3
PDB

GoogleScholar
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PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363502
PNG
(US9850257, Example 9)
Show SMILES Cc1noc(C)c1-c1cc(Br)c2cnn3C(COc1c23)c1ccccc1
Show InChI InChI=1/C20H16BrN3O2/c1-11-18(12(2)26-23-11)14-8-16(21)15-9-22-24-17(10-25-20(14)19(15)24)13-6-4-3-5-7-13/h3-9,17H,10H2,1-2H3
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363498
PNG
(US9850257, Example 5)
Show SMILES Cc1noc(C)c1-c1ccc2c3c1OCC(c1ccccn1)n3[nH]c2=O
Show InChI InChI=1/C19H16N4O3/c1-10-16(11(2)26-22-10)12-6-7-13-17-18(12)25-9-15(23(17)21-19(13)24)14-5-3-4-8-20-14/h3-8,15H,9H2,1-2H3,(H,21,24)
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM50158618
PNG
(CHEMBL3787341 | US9850257, Example 11)
Show SMILES Cc1noc(C)c1-c1ccc2c3c1OCC(c1cccnc1)n3n(C)c2=O
Show InChI InChI=1/C20H18N4O3/c1-11-17(12(2)27-22-11)14-6-7-15-18-19(14)26-10-16(13-5-4-8-21-9-13)24(18)23(3)20(15)25/h4-9,16H,10H2,1-3H3
PDB

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US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363494
PNG
(US9850257, Example 1)
Show SMILES Cc1noc(C)c1-c1ccc2c3c1OCC(c1ccccc1)n3[nH]c2=O
Show InChI InChI=1/C20H17N3O3/c1-11-17(12(2)26-22-11)14-8-9-15-18-19(14)25-10-16(23(18)21-20(15)24)13-6-4-3-5-7-13/h3-9,16H,10H2,1-2H3,(H,21,24)
PDB

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PC cid
PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363495
PNG
(9-(3,5-Dimethylisoxazol-4-yl)-5-methyl-3-phenyl-2,...)
Show SMILES Cc1noc(C)c1-c1ccc2c3c1OCC(c1ccccc1)n3n(C)c2=O
Show InChI InChI=1/C21H19N3O3/c1-12-18(13(2)27-22-12)15-9-10-16-19-20(15)26-11-17(14-7-5-4-6-8-14)24(19)23(3)21(16)25/h4-10,17H,11H2,1-3H3
PDB

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PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363497
PNG
(US9850257, Example 4)
Show SMILES Cc1noc(C)c1-c1ccc2cnn3C(COc1c23)c1ccccc1
Show InChI InChI=1/C20H17N3O2/c1-12-18(13(2)25-22-12)16-9-8-15-10-21-23-17(11-24-20(16)19(15)23)14-6-4-3-5-7-14/h3-10,17H,11H2,1-2H3
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363501
PNG
(US9850257, Example 8)
Show SMILES Cc1noc(C)c1-c1ccc2cnn3C(COc1c23)c1ccccn1
Show InChI InChI=1/C19H16N4O2/c1-11-17(12(2)25-22-11)14-7-6-13-9-21-23-16(10-24-19(14)18(13)23)15-5-3-4-8-20-15/h3-9,16H,10H2,1-2H3
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363495
PNG
(9-(3,5-Dimethylisoxazol-4-yl)-5-methyl-3-phenyl-2,...)
Show SMILES Cc1noc(C)c1-c1ccc2c3c1OCC(c1ccccc1)n3n(C)c2=O
Show InChI InChI=1/C21H19N3O3/c1-12-18(13(2)27-22-12)15-9-10-16-19-20(15)26-11-17(14-7-5-4-6-8-14)24(19)23(3)21(16)25/h4-10,17H,11H2,1-3H3
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363496
PNG
(9-(3,5-Dimethylisoxazol-4-yl)-6-methoxy-3-phenyl-2...)
Show SMILES COc1nn2C(COc3c(ccc1c23)-c1c(C)noc1C)c1ccccc1
Show InChI InChI=1/C21H19N3O3/c1-12-18(13(2)27-23-12)15-9-10-16-19-20(15)26-11-17(14-7-5-4-6-8-14)24(19)22-21(16)25-3/h4-10,17H,11H2,1-3H3
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363496
PNG
(9-(3,5-Dimethylisoxazol-4-yl)-6-methoxy-3-phenyl-2...)
Show SMILES COc1nn2C(COc3c(ccc1c23)-c1c(C)noc1C)c1ccccc1
Show InChI InChI=1/C21H19N3O3/c1-12-18(13(2)27-23-12)15-9-10-16-19-20(15)26-11-17(14-7-5-4-6-8-14)24(19)22-21(16)25-3/h4-10,17H,11H2,1-3H3
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363503
PNG
(US9850257, Example 10)
Show SMILES Cc1noc(C)c1-c1ccc2c3c1OCC(c1cccnc1)n3[nH]c2=O
Show InChI InChI=1/C19H16N4O3/c1-10-16(11(2)26-22-10)13-5-6-14-17-18(13)25-9-15(23(17)21-19(14)24)12-4-3-7-20-8-12/h3-8,15H,9H2,1-2H3,(H,21,24)
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363500
PNG
(9-(3,5-Dimethylisoxazol-4-yl)-6-methoxy-3-pyridin-...)
Show SMILES COc1nn2C(COc3c(ccc1c23)-c1c(C)noc1C)c1ccccn1
Show InChI InChI=1/C20H18N4O3/c1-11-17(12(2)27-23-11)13-7-8-14-18-19(13)26-10-16(15-6-4-5-9-21-15)24(18)22-20(14)25-3/h4-9,16H,10H2,1-3H3
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363494
PNG
(US9850257, Example 1)
Show SMILES Cc1noc(C)c1-c1ccc2c3c1OCC(c1ccccc1)n3[nH]c2=O
Show InChI InChI=1/C20H17N3O3/c1-11-17(12(2)26-22-11)14-8-9-15-18-19(14)25-10-16(23(18)21-20(15)24)13-6-4-3-5-7-13/h3-9,16H,10H2,1-2H3,(H,21,24)
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363497
PNG
(US9850257, Example 4)
Show SMILES Cc1noc(C)c1-c1ccc2cnn3C(COc1c23)c1ccccc1
Show InChI InChI=1/C20H17N3O2/c1-12-18(13(2)25-22-12)16-9-8-15-10-21-23-17(11-24-20(16)19(15)23)14-6-4-3-5-7-14/h3-10,17H,11H2,1-2H3
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363499
PNG
(9-(3,5-Dimethylisoxazol-4-yl)-5-methyl-3-pyridin-2...)
Show SMILES Cc1noc(C)c1-c1ccc2c3c1OCC(c1ccccn1)n3n(C)c2=O
Show InChI InChI=1/C20H18N4O3/c1-11-17(12(2)27-22-11)13-7-8-14-18-19(13)26-10-16(15-6-4-5-9-21-15)24(18)23(3)20(14)25/h4-9,16H,10H2,1-3H3
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363500
PNG
(9-(3,5-Dimethylisoxazol-4-yl)-6-methoxy-3-pyridin-...)
Show SMILES COc1nn2C(COc3c(ccc1c23)-c1c(C)noc1C)c1ccccn1
Show InChI InChI=1/C20H18N4O3/c1-11-17(12(2)27-23-11)13-7-8-14-18-19(13)26-10-16(15-6-4-5-9-21-15)24(18)22-20(14)25-3/h4-9,16H,10H2,1-3H3
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363501
PNG
(US9850257, Example 8)
Show SMILES Cc1noc(C)c1-c1ccc2cnn3C(COc1c23)c1ccccn1
Show InChI InChI=1/C19H16N4O2/c1-11-17(12(2)25-22-11)14-7-6-13-9-21-23-16(10-24-19(14)18(13)23)15-5-3-4-8-20-15/h3-9,16H,10H2,1-2H3
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM50158618
PNG
(CHEMBL3787341 | US9850257, Example 11)
Show SMILES Cc1noc(C)c1-c1ccc2c3c1OCC(c1cccnc1)n3n(C)c2=O
Show InChI InChI=1/C20H18N4O3/c1-11-17(12(2)27-22-11)14-6-7-15-18-19(14)26-10-16(13-5-4-8-21-9-13)24(18)23(3)20(15)25/h4-9,16H,10H2,1-3H3
PDB

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UniChem

Similars

US Patent
n/an/a<200n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363498
PNG
(US9850257, Example 5)
Show SMILES Cc1noc(C)c1-c1ccc2c3c1OCC(c1ccccn1)n3[nH]c2=O
Show InChI InChI=1/C19H16N4O3/c1-10-16(11(2)26-22-10)12-6-7-13-17-18(12)25-9-15(23(17)21-19(13)24)14-5-3-4-8-20-14/h3-8,15H,9H2,1-2H3,(H,21,24)
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a 600n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363508
PNG
(US9850257, Example 13)
Show SMILES Cc1noc(C)c1-c1cc(F)c2nnn3C(COc1c23)c1cccnc1
Show InChI InChI=1/C18H14FN5O2/c1-9-15(10(2)26-22-9)12-6-13(19)16-17-18(12)25-8-14(24(17)23-21-16)11-4-3-5-20-7-11/h3-7,14H,8H2,1-2H3
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a 600n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363503
PNG
(US9850257, Example 10)
Show SMILES Cc1noc(C)c1-c1ccc2c3c1OCC(c1cccnc1)n3[nH]c2=O
Show InChI InChI=1/C19H16N4O3/c1-10-16(11(2)26-22-10)13-5-6-14-17-18(13)25-9-15(23(17)21-19(14)24)12-4-3-7-20-8-12/h3-8,15H,9H2,1-2H3,(H,21,24)
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a 600n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363502
PNG
(US9850257, Example 9)
Show SMILES Cc1noc(C)c1-c1cc(Br)c2cnn3C(COc1c23)c1ccccc1
Show InChI InChI=1/C20H16BrN3O2/c1-11-18(12(2)26-23-11)14-8-16(21)15-9-22-24-17(10-25-20(14)19(15)24)13-6-4-3-5-7-13/h3-9,17H,10H2,1-2H3
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a 600n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
Bromodomain containing 4


(Homo sapiens (Human))
BDBM363508
PNG
(US9850257, Example 13)
Show SMILES Cc1noc(C)c1-c1cc(F)c2nnn3C(COc1c23)c1cccnc1
Show InChI InChI=1/C18H14FN5O2/c1-9-15(10(2)26-22-9)12-6-13(19)16-17-18(12)25-8-14(24(17)23-21-16)11-4-3-5-20-7-11/h3-7,14H,8H2,1-2H3
PDB

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a>1.00E+3n/an/an/an/an/an/a



Incyte Corporation; Incyte Holdings Corporation

US Patent


Assay Description
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...


US Patent US9850257 (2017)

More data for this
Ligand-Target Pair
* indicates data uncertainty>20%