Compile Data Set for Download or QSAR
maximum 50k data
Found 331 Enz. Inhib. hit(s) with all data for entry = 2449
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366233(US9873693, Compound 156)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366234(US9873693, Compound 157)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366236(US9873693, Compound 159)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366237(US9873693, Compound 160)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366238(US9873693, Compound 161)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366328(US9873693, Compound 255)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366330(US9873693, Compound 257)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366331(US9873693, Compound 258)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366332(US9873693, Compound 259)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366183(US9873693, Compound 106 | US9873693, Compound 260)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366335(US9873693, Compound 262)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366336(US9873693, Compound 263)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366186(US9873693, Compound 109 | US9873693, Compound 264)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366098(US9873693, Compound 21)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366099(US9873693, Compound 22)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366100(US9873693, Compound 23)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366101(US9873693, Compound 24)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366102(US9873693, Compound 25)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366103(US9873693, Compound 26)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366216(US9873693, Compound 139)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366217(US9873693, Compound 140)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366218(US9873693, Compound 141)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366219(US9873693, Compound 142)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366220(US9873693, Compound 143)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM50361645(CHEMBL1234429 | US9873693, Compound 144)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366222(US9873693, Compound 145)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366223(US9873693, Compound 146)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366092(US9873693, Compound 15 | US9873693, Compound 234)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366312(US9873693, Compound 237)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366313(US9873693, Compound 238)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366314(US9873693, Compound 239)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366104(US9873693, Compound 27)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366105(US9873693, Compound 28)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366106(US9873693, Compound 29)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366107(US9873693, Compound 30)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366108(US9873693, Compound 31)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366109(US9873693, Compound 32)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366110(US9873693, Compound 33)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366111(US9873693, Compound 34)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366140(US9873693, Compound 63)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366141(US9873693, Compound 64)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366142(US9873693, Compound 65)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366143(US9873693, Compound 66)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366144(US9873693, Compound 67)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366145(US9873693, Compound 68)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366146(US9873693, Compound 69)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366147(US9873693, Compound 70)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366148(US9873693, Compound 71)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366224(US9873693, Compound 147)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Sunesis Pharmaceuticals

US Patent
LigandPNGBDBM366225(US9873693, Compound 148)
Affinity DataIC50: <500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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