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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| RET Kinase (aa658-end) (Homo sapiens (Human)) | BDBM376119 (N-(2-(dimethylamino)ethyl)-3-(2-(4-(4-ethoxy-6-oxo...) | PDB GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED US Patent | Assay Description Human RET kinase cytoplasmic domain (amino acids 658-1114 of accession number NP_000314.1) was expressed as an N-terminal GST-fusion protein using a ... | US Patent US9918974 (2018) | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| RET Kinase (aa658-end) (Homo sapiens (Human)) | BDBM376389 (N-(3-(2-(dimethylamino)ethoxy)-5-(trifluoromethyl)...) | PDB GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED US Patent | Assay Description Human RET kinase cytoplasmic domain (amino acids 658-1114 of accession number NP_000314.1) was expressed as an N-terminal GST-fusion protein using a ... | US Patent US9918974 (2018) | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
