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Patent code US9969726

Compile Data Set for Download or QSAR

Found 724 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393729
PNG
(US10597367, Example 19 | US9969726, Example 19)
Show SMILES COc1cc(ccc1F)-c1cccc(c1)-c1csc(n1)-c1ccccc1
Show InChI InChI=1S/C22H16FNOS/c1-25-21-13-17(10-11-19(21)23)16-8-5-9-18(12-16)20-14-26-22(24-20)15-6-3-2-4-7-15/h2-14H,1H3
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n/an/an/an/a 1.55E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393729
PNG
(US10597367, Example 19 | US9969726, Example 19)
Show SMILES COc1cc(ccc1F)-c1cccc(c1)-c1csc(n1)-c1ccccc1
Show InChI InChI=1S/C22H16FNOS/c1-25-21-13-17(10-11-19(21)23)16-8-5-9-18(12-16)20-14-26-22(24-20)15-6-3-2-4-7-15/h2-14H,1H3
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n/an/an/an/a>1.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393729
PNG
(US10597367, Example 19 | US9969726, Example 19)
Show SMILES COc1cc(ccc1F)-c1cccc(c1)-c1csc(n1)-c1ccccc1
Show InChI InChI=1S/C22H16FNOS/c1-25-21-13-17(10-11-19(21)23)16-8-5-9-18(12-16)20-14-26-22(24-20)15-6-3-2-4-7-15/h2-14H,1H3
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n/an/an/an/a>1.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393730
PNG
(US9969726, Example 20)
Show SMILES O\N=C/c1cc(ccc1F)-c1cccc(c1)-c1csc(n1)-c1ccccc1
Show InChI InChI=1S/C22H15FN2OS/c23-20-10-9-17(12-19(20)13-24-26)16-7-4-8-18(11-16)21-14-27-22(25-21)15-5-2-1-3-6-15/h1-14,26H/b24-13-
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n/an/an/an/a>3.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393737
PNG
(US10597367, Example 27 | US9969726, Example 27)
Show SMILES Fc1ccc(cc1)-c1csc(n1)-c1ccccc1
Show InChI InChI=1S/C15H10FNS/c16-13-8-6-11(7-9-13)14-10-18-15(17-14)12-4-2-1-3-5-12/h1-10H
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n/an/an/an/a>3.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393737
PNG
(US10597367, Example 27 | US9969726, Example 27)
Show SMILES Fc1ccc(cc1)-c1csc(n1)-c1ccccc1
Show InChI InChI=1S/C15H10FNS/c16-13-8-6-11(7-9-13)14-10-18-15(17-14)12-4-2-1-3-5-12/h1-10H
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n/an/an/an/a>3.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393737
PNG
(US10597367, Example 27 | US9969726, Example 27)
Show SMILES Fc1ccc(cc1)-c1csc(n1)-c1ccccc1
Show InChI InChI=1S/C15H10FNS/c16-13-8-6-11(7-9-13)14-10-18-15(17-14)12-4-2-1-3-5-12/h1-10H
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n/an/an/an/a>3.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393742
PNG
(US10597367, Example 32 | US9969726, Example 32)
Show SMILES c1sc(nc1-c1cccc(c1)-c1ccccc1)-c1ccc2ccccc2c1
Show InChI InChI=1S/C25H17NS/c1-2-7-18(8-3-1)21-11-6-12-22(15-21)24-17-27-25(26-24)23-14-13-19-9-4-5-10-20(19)16-23/h1-17H
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n/an/an/an/a 4.98E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393743
PNG
(US10597367, Example 33 | US9969726, Example 33)
Show SMILES OC(=O)c1cccc(c1)-c1nc(cs1)-c1cccc(c1)-c1ccccc1
Show InChI InChI=1S/C22H15NO2S/c24-22(25)19-11-5-10-18(13-19)21-23-20(14-26-21)17-9-4-8-16(12-17)15-6-2-1-3-7-15/h1-14H,(H,24,25)
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n/an/an/an/a 4.83E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393745
PNG
(US10597367, Example 35 | US9969726, Example 35)
Show SMILES Clc1ccc(cn1)-c1nc(cs1)-c1cccc(c1)-c1ccccc1
Show InChI InChI=1S/C20H13ClN2S/c21-19-10-9-17(12-22-19)20-23-18(13-24-20)16-8-4-7-15(11-16)14-5-2-1-3-6-14/h1-13H
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n/an/an/an/a 830n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393746
PNG
(US10597367, Example 36 | US9969726, Example 36)
Show SMILES C(=C/c1ccccc1)\c1nc(cs1)-c1cccc(c1)-c1ccccc1
Show InChI InChI=1S/C23H17NS/c1-3-8-18(9-4-1)14-15-23-24-22(17-25-23)21-13-7-12-20(16-21)19-10-5-2-6-11-19/h1-17H/b15-14+
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n/an/an/an/a 3.47E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393748
PNG
(US10597367, Example 38 | US9969726, Example 38)
Show SMILES Fc1ccc(cc1)-c1cccc(c1)-c1nsc(n1)-c1ccccc1
Show InChI InChI=1S/C20H13FN2S/c21-18-11-9-14(10-12-18)16-7-4-8-17(13-16)19-22-20(24-23-19)15-5-2-1-3-6-15/h1-13H
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n/an/an/an/a 100n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393748
PNG
(US10597367, Example 38 | US9969726, Example 38)
Show SMILES Fc1ccc(cc1)-c1cccc(c1)-c1nsc(n1)-c1ccccc1
Show InChI InChI=1S/C20H13FN2S/c21-18-11-9-14(10-12-18)16-7-4-8-17(13-16)19-22-20(24-23-19)15-5-2-1-3-6-15/h1-13H
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n/an/an/an/a 520n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393749
PNG
(US10597367, Example 39 | US9969726, Example 39)
Show SMILES c1ccc(cc1)-c1nc(ns1)-c1cccc(c1)-c1ccccc1
Show InChI InChI=1S/C20H14N2S/c1-3-8-15(9-4-1)17-12-7-13-18(14-17)19-21-20(23-22-19)16-10-5-2-6-11-16/h1-14H
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n/an/an/an/a 50n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393753
PNG
(BDBM437895 | US9969726, Example 43)
Show SMILES Fc1cccc(c1)-c1cccc(c1)-c1nsc(n1)-c1ccoc1
Show InChI InChI=1S/C18H11FN2OS/c19-16-6-2-4-13(10-16)12-3-1-5-14(9-12)17-20-18(23-21-17)15-7-8-22-11-15/h1-11H
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n/an/an/an/a 110n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393754
PNG
(US10597367, Example 44 | US9969726, Example 44)
Show SMILES OC(=O)c1cccc(c1)-c1cccc(c1)-c1cc(sn1)-c1ccccc1
Show InChI InChI=1S/C22H15NO2S/c24-22(25)19-11-5-9-17(13-19)16-8-4-10-18(12-16)20-14-21(26-23-20)15-6-2-1-3-7-15/h1-14H,(H,24,25)
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n/an/an/an/a 180n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393755
PNG
(US10597367, Example 45 | US9969726, Example 45)
Show SMILES Fc1ccc(cc1)-c1cccc(c1)-c1csc(c1)-c1ccccc1
Show InChI InChI=1S/C22H15FS/c23-21-11-9-16(10-12-21)18-7-4-8-19(13-18)20-14-22(24-15-20)17-5-2-1-3-6-17/h1-15H
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n/an/an/an/a>1.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393756
PNG
(US9969726, Example 46)
Show SMILES OC(=O)c1cccc(c1)-c1cccc(c1)-c1coc(n1)-c1ccccc1
Show InChI InChI=1S/C22H15NO3/c24-22(25)19-11-5-9-17(13-19)16-8-4-10-18(12-16)20-14-26-21(23-20)15-6-2-1-3-7-15/h1-14H,(H,24,25)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393759
PNG
(US10597367, Example 49 | US9969726, Example 49)
Show SMILES c1c(noc1-c1ccccc1)-c1cccc(c1)-c1ccccc1
Show InChI InChI=1S/C21H15NO/c1-3-8-16(9-4-1)18-12-7-13-19(14-18)20-15-21(23-22-20)17-10-5-2-6-11-17/h1-15H
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n/an/an/an/a>3.00E+4n/an/an/an/a



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US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393762
PNG
(US10597367, Example 51 | US9969726, Example 51)
Show SMILES Fc1ccc(cc1)-c1cccc(c1)-c1nc(-c2ccccc2)n(n1)-c1ccccc1
Show InChI InChI=1S/C26H18FN3/c27-23-16-14-19(15-17-23)21-10-7-11-22(18-21)25-28-26(20-8-3-1-4-9-20)30(29-25)24-12-5-2-6-13-24/h1-18H
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Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393764
PNG
(US10597367, Example 53 | US9969726, Example 53)
Show SMILES c1csc(c1)-c1nc(nn1-c1ccccc1)-c1cccc(c1)-c1ccccc1
Show InChI InChI=1S/C24H17N3S/c1-3-9-18(10-4-1)19-11-7-12-20(17-19)23-25-24(22-15-8-16-28-22)27(26-23)21-13-5-2-6-14-21/h1-17H
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n/an/an/an/a>1.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393764
PNG
(US10597367, Example 53 | US9969726, Example 53)
Show SMILES c1csc(c1)-c1nc(nn1-c1ccccc1)-c1cccc(c1)-c1ccccc1
Show InChI InChI=1S/C24H17N3S/c1-3-9-18(10-4-1)19-11-7-12-20(17-19)23-25-24(22-15-8-16-28-22)27(26-23)21-13-5-2-6-14-21/h1-17H
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n/an/an/an/a 4.29E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393768
PNG
(US10597367, Example 57 | US9969726, Example 57)
Show SMILES c1ccc(cc1)-c1nc(nn1-c1cccc2ccccc12)-c1cccc(c1)-c1ccccc1
Show InChI InChI=1S/C30H21N3/c1-3-11-22(12-4-1)25-17-9-18-26(21-25)29-31-30(24-14-5-2-6-15-24)33(32-29)28-20-10-16-23-13-7-8-19-27(23)28/h1-21H
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n/an/an/an/a>1.00E+4n/an/an/an/a



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US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393768
PNG
(US10597367, Example 57 | US9969726, Example 57)
Show SMILES c1ccc(cc1)-c1nc(nn1-c1cccc2ccccc12)-c1cccc(c1)-c1ccccc1
Show InChI InChI=1S/C30H21N3/c1-3-11-22(12-4-1)25-17-9-18-26(21-25)29-31-30(24-14-5-2-6-15-24)33(32-29)28-20-10-16-23-13-7-8-19-27(23)28/h1-21H
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n/an/an/an/a>1.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393760
PNG
(US10597367, Example 60 | US9969726, Example 49A | ...)
Show SMILES c1ccc(cc1)-c1nc(nn1-c1ccccc1)-c1cccc(c1)-c1ccccc1
Show InChI InChI=1S/C26H19N3/c1-4-11-20(12-5-1)22-15-10-16-23(19-22)25-27-26(21-13-6-2-7-14-21)29(28-25)24-17-8-3-9-18-24/h1-19H
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n/an/an/an/a>1.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393776
PNG
(US10597367, Example 65 | US9969726, Example 65)
Show SMILES c1ccc(cc1)-c1nc(n[nH]1)-c1cccc(c1)-c1ccccc1
Show InChI InChI=1S/C20H15N3/c1-3-8-15(9-4-1)17-12-7-13-18(14-17)20-21-19(22-23-20)16-10-5-2-6-11-16/h1-14H,(H,21,22,23)
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n/an/an/an/a>3.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393776
PNG
(US10597367, Example 65 | US9969726, Example 65)
Show SMILES c1ccc(cc1)-c1nc(n[nH]1)-c1cccc(c1)-c1ccccc1
Show InChI InChI=1S/C20H15N3/c1-3-8-15(9-4-1)17-12-7-13-18(14-17)20-21-19(22-23-20)16-10-5-2-6-11-16/h1-14H,(H,21,22,23)
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n/an/an/an/a>3.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393777
PNG
(US10597367, Example 66 | US9969726, Example 66)
Show SMILES OC(=O)c1cccc(c1)-c1cccc(c1)-c1nc(nn1-c1ccccc1)-c1ccccc1
Show InChI InChI=1S/C27H19N3O2/c31-27(32)23-14-8-12-21(18-23)20-11-7-13-22(17-20)26-28-25(19-9-3-1-4-10-19)29-30(26)24-15-5-2-6-16-24/h1-18H,(H,31,32)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393779
PNG
(US10597367, Example 68 | US9969726, Example 68)
Show SMILES OC(=O)c1cccc(c1)-c1cccc(c1)-c1cc([nH]n1)-c1ccccc1
Show InChI InChI=1S/C22H16N2O2/c25-22(26)19-11-5-9-17(13-19)16-8-4-10-18(12-16)21-14-20(23-24-21)15-6-2-1-3-7-15/h1-14H,(H,23,24)(H,25,26)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393780
PNG
(US10597367, Example 69 | US9969726, Example 69)
Show SMILES OC(=O)c1cccc(c1)-c1cccc(c1)-c1nc(cc(n1)C(F)(F)F)-c1ccc(nc1)C(F)(F)F
Show InChI InChI=1S/C24H13F6N3O2/c25-23(26,27)19-8-7-17(12-31-19)18-11-20(24(28,29)30)33-21(32-18)15-5-1-3-13(9-15)14-4-2-6-16(10-14)22(34)35/h1-12H,(H,34,35)
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n/an/an/an/a 110n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393784
PNG
(US10597367, Example 73 | US9969726, Example 73)
Show SMILES OC(=O)c1cc(ccc1F)-c1cccc(c1)-c1nc(cc(n1)C(F)(F)F)-c1ccc(nc1)C(F)(F)F
Show InChI InChI=1S/C24H12F7N3O2/c25-17-6-4-13(9-16(17)22(35)36)12-2-1-3-14(8-12)21-33-18(10-20(34-21)24(29,30)31)15-5-7-19(32-11-15)23(26,27)28/h1-11H,(H,35,36)
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n/an/an/an/a 1.18E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393787
PNG
(US10597367, Example 76 | US9969726, Example 76)
Show SMILES OC(=O)c1cc(F)cc(c1)-c1cccc(c1)-c1nc(cc(n1)C(F)(F)F)-c1ccc(nc1)C(F)(F)F
Show InChI InChI=1S/C24H12F7N3O2/c25-17-8-15(7-16(9-17)22(35)36)12-2-1-3-13(6-12)21-33-18(10-20(34-21)24(29,30)31)14-4-5-19(32-11-14)23(26,27)28/h1-11H,(H,35,36)
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n/an/an/an/a 1.61E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393788
PNG
(US10597367, Example 77 | US9969726, Example 77)
Show SMILES COc1ccc(cc1-c1cccc(c1)-c1nc(cc(n1)C(F)(F)F)-c1ccc(nc1)C(F)(F)F)C(O)=O
Show InChI InChI=1S/C25H15F6N3O3/c1-37-19-7-5-15(23(35)36)10-17(19)13-3-2-4-14(9-13)22-33-18(11-21(34-22)25(29,30)31)16-6-8-20(32-12-16)24(26,27)28/h2-12H,1H3,(H,35,36)
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n/an/an/an/a 1.70E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393789
PNG
(US10597367, Example 78 | US9969726, Example 78)
Show SMILES OC(=O)c1ccc(c(Cl)c1)-c1cccc(c1)-c1nc(cc(n1)C(F)(F)F)-c1ccc(nc1)C(F)(F)F
Show InChI InChI=1S/C24H12ClF6N3O2/c25-17-9-14(22(35)36)4-6-16(17)12-2-1-3-13(8-12)21-33-18(10-20(34-21)24(29,30)31)15-5-7-19(32-11-15)23(26,27)28/h1-11H,(H,35,36)
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n/an/an/an/a 6.32E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393797
PNG
(US10597367, Example 86 | US9969726, Example 86)
Show SMILES OC(=O)c1cc(ccc1F)-c1cccc(c1)-c1nc(cc(n1)C(F)(F)F)-c1ccccc1
Show InChI InChI=1S/C24H14F4N2O2/c25-19-10-9-16(12-18(19)23(31)32)15-7-4-8-17(11-15)22-29-20(14-5-2-1-3-6-14)13-21(30-22)24(26,27)28/h1-13H,(H,31,32)
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n/an/an/an/a 120n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393801
PNG
(US10597367, Example 89 | US9969726, Example 89)
Show SMILES OC(=O)c1cc(F)cc(c1)-c1cccc(c1)-c1nc(cc(n1)C(F)(F)F)-c1ccco1
Show InChI InChI=1S/C22H12F4N2O3/c23-16-9-14(8-15(10-16)21(29)30)12-3-1-4-13(7-12)20-27-17(18-5-2-6-31-18)11-19(28-20)22(24,25)26/h1-11H,(H,29,30)
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n/an/an/an/a 2.25E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393803
PNG
(US10597367, Example 91 | US9969726, Example 91)
Show SMILES Cc1ccccc1-c1cc(nc(n1)-c1cccc(c1)-c1ccc(F)c(c1)C(O)=O)C(F)(F)F
Show InChI InChI=1S/C25H16F4N2O2/c1-14-5-2-3-8-18(14)21-13-22(25(27,28)29)31-23(30-21)17-7-4-6-15(11-17)16-9-10-20(26)19(12-16)24(32)33/h2-13H,1H3,(H,32,33)
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n/an/an/an/a 1.52E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393804
PNG
(US10597367, Example 92 | US9969726, Example 92)
Show SMILES Cc1cccc(c1)-c1cc(nc(n1)-c1cccc(c1)-c1ccc(F)c(c1)C(O)=O)C(F)(F)F
Show InChI InChI=1S/C25H16F4N2O2/c1-14-4-2-6-17(10-14)21-13-22(25(27,28)29)31-23(30-21)18-7-3-5-15(11-18)16-8-9-20(26)19(12-16)24(32)33/h2-13H,1H3,(H,32,33)
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n/an/an/an/a 2.79E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393804
PNG
(US10597367, Example 92 | US9969726, Example 92)
Show SMILES Cc1cccc(c1)-c1cc(nc(n1)-c1cccc(c1)-c1ccc(F)c(c1)C(O)=O)C(F)(F)F
Show InChI InChI=1S/C25H16F4N2O2/c1-14-4-2-6-17(10-14)21-13-22(25(27,28)29)31-23(30-21)18-7-3-5-15(11-18)16-8-9-20(26)19(12-16)24(32)33/h2-13H,1H3,(H,32,33)
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n/an/an/an/a 400n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393807
PNG
(US10597367, Example 95 | US9969726, Example 95)
Show SMILES OC(=O)c1cc(ccc1F)-c1cccc(c1)-c1nc(\C=C\c2ccccc2)cc(n1)C(F)(F)F
Show InChI InChI=1S/C26H16F4N2O2/c27-22-12-10-18(14-21(22)25(33)34)17-7-4-8-19(13-17)24-31-20(15-23(32-24)26(28,29)30)11-9-16-5-2-1-3-6-16/h1-15H,(H,33,34)/b11-9+
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n/an/an/an/a>1.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393809
PNG
(US10597367, Example 97 | US9969726, Example 97)
Show SMILES OC(=O)c1cc(ccc1F)-c1cccc(c1)-c1nc(cc(n1)C(F)(F)F)-c1cccnc1F
Show InChI InChI=1S/C23H12F5N3O2/c24-17-7-6-13(10-16(17)22(32)33)12-3-1-4-14(9-12)21-30-18(11-19(31-21)23(26,27)28)15-5-2-8-29-20(15)25/h1-11H,(H,32,33)
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n/an/an/an/a 1.71E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393812
PNG
(US10597367, Example 100 | US9969726, Example 100)
Show SMILES OC(=O)c1cc(ccc1F)-c1cccc(c1)-c1nc(cc(n1)C(F)(F)F)-c1ccccc1F
Show InChI InChI=1S/C24H13F5N2O2/c25-18-7-2-1-6-16(18)20-12-21(24(27,28)29)31-22(30-20)15-5-3-4-13(10-15)14-8-9-19(26)17(11-14)23(32)33/h1-12H,(H,32,33)
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n/an/an/an/a 1.21E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393816
PNG
(US10597367, Example 104 | US9969726, Example 104)
Show SMILES OC(=O)c1cc(F)cc(c1)-c1cccc(c1)-c1nc(cc(n1)C(F)(F)F)-c1ccccc1
Show InChI InChI=1S/C24H14F4N2O2/c25-19-11-17(10-18(12-19)23(31)32)15-7-4-8-16(9-15)22-29-20(14-5-2-1-3-6-14)13-21(30-22)24(26,27)28/h1-13H,(H,31,32)
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n/an/an/an/a 1.44E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393819
PNG
(US10597367, Example 107 | US9969726, Example 107)
Show SMILES OC(=O)c1cc(ccc1F)-c1cccc(c1)-c1nc(cc(n1)C(F)(F)F)-c1sccc1Cl
Show InChI InChI=1S/C22H11ClF4N2O2S/c23-15-6-7-32-19(15)17-10-18(22(25,26)27)29-20(28-17)13-3-1-2-11(8-13)12-4-5-16(24)14(9-12)21(30)31/h1-10H,(H,30,31)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393820
PNG
(US10597367, Example 108 | US9969726, Example 108)
Show SMILES OC(=O)c1cc(ccc1F)-c1cccc(c1)-c1nc(cc(n1)C(F)(F)F)-c1ccc(cc1)C(F)(F)F
Show InChI InChI=1S/C25H13F7N2O2/c26-19-9-6-15(11-18(19)23(35)36)14-2-1-3-16(10-14)22-33-20(12-21(34-22)25(30,31)32)13-4-7-17(8-5-13)24(27,28)29/h1-12H,(H,35,36)
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US Patent
n/an/an/an/a 150n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393821
PNG
(US10597367, Example 109 | US9969726, Example 109)
Show SMILES OC(=O)c1cc(ccc1F)-c1cccc(c1)-c1nc(cc(n1)C(F)(F)F)-c1nccs1
Show InChI InChI=1S/C21H11F4N3O2S/c22-15-5-4-12(9-14(15)20(29)30)11-2-1-3-13(8-11)18-27-16(19-26-6-7-31-19)10-17(28-18)21(23,24)25/h1-10H,(H,29,30)
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US Patent
n/an/an/an/a 2.13E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393823
PNG
(US10597367, Example 111 | US9969726, Example 111)
Show SMILES Cc1noc(C)c1-c1cc(nc(n1)-c1cccc(c1)-c1ccc(F)c(c1)C(O)=O)C(F)(F)F
Show InChI InChI=1S/C23H15F4N3O3/c1-11-20(12(2)33-30-11)18-10-19(23(25,26)27)29-21(28-18)15-5-3-4-13(8-15)14-6-7-17(24)16(9-14)22(31)32/h3-10H,1-2H3,(H,31,32)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393832
PNG
(US10597367, Example 120 | US9969726, Example 120)
Show SMILES COc1ccc(cn1)-c1cc(nc(n1)-c1cccc(c1)-c1ccc(F)c(c1)C(O)=O)C(F)(F)F
Show InChI InChI=1S/C24H15F4N3O3/c1-34-21-8-6-16(12-29-21)19-11-20(24(26,27)28)31-22(30-19)15-4-2-3-13(9-15)14-5-7-18(25)17(10-14)23(32)33/h2-12H,1H3,(H,32,33)
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n/an/an/an/a 1.41E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 2


(Rattus norvegicus)
BDBM393825
PNG
(US10597367, Example 113 | US9969726, Example 113 |...)
Show SMILES OC(=O)c1cc(F)cc(c1)-c1cccc(c1)-c1nc(cc(n1)C(F)(F)F)-c1ccoc1
Show InChI InChI=1S/C22H12F4N2O3/c23-17-8-15(7-16(9-17)21(29)30)12-2-1-3-13(6-12)20-27-18(14-4-5-31-11-14)10-19(28-20)22(24,25)26/h1-11H,(H,29,30)
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n/an/an/an/a 310n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 3


(Rattus norvegicus (Rat))
BDBM393825
PNG
(US10597367, Example 113 | US9969726, Example 113 |...)
Show SMILES OC(=O)c1cc(F)cc(c1)-c1cccc(c1)-c1nc(cc(n1)C(F)(F)F)-c1ccoc1
Show InChI InChI=1S/C22H12F4N2O3/c23-17-8-15(7-16(9-17)21(29)30)12-2-1-3-13(6-12)20-27-18(14-4-5-31-11-14)10-19(28-20)22(24,25)26/h1-11H,(H,29,30)
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US Patent
n/an/an/an/a 2.21E+3n/an/an/an/a



Sanford-Burnham Medical Research Institute

US Patent


Assay Description
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...


US Patent US9969726 (2018)


BindingDB Entry DOI: 10.7270/Q2RX9FDX
More data for this
Ligand-Target Pair
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* indicates data uncertainty>20%