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Found 11 Enz. Inhib. hit(s) with all data for entry = 2729
TargetAdenosine receptor A2a(GUINEA PIG)
Gilead Sciences

US Patent
LigandPNGBDBM377134(Ethyl 1-{9-[(4S,2R,3R,5R)-3,4-dihydroxy-5-(hydroxy...)
Affinity DataKi:  505nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(GUINEA PIG)
Gilead Sciences

US Patent
LigandPNGBDBM377143((1-{9-[(4S,2R,3R,5R)-3,4-dihydroxy-5-(hydroxymethy...)
Affinity DataKi:  505nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(GUINEA PIG)
Gilead Sciences

US Patent
LigandPNGBDBM377142(1-{9-[(4S,2R,3R,5R)-3,4-dihydroxy-5-(hydroxymethyl...)
Affinity DataKi:  505nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(GUINEA PIG)
Gilead Sciences

US Patent
LigandPNGBDBM377141((1-{9-[(4S,2R,3R,5R)-3,4-dihydroxy-5-(hydrozymethy...)
Affinity DataKi:  505nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(GUINEA PIG)
Gilead Sciences

US Patent
LigandPNGBDBM377140((1-{9-[(4S,2R,3R,5R)-3,4-dihydroxy-5-(hydroxymethy...)
Affinity DataKi:  505nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(GUINEA PIG)
Gilead Sciences

US Patent
LigandPNGBDBM377144((1-{9-[(4S,2R,3R,5R)-3,4-dihydroxy-5-(hydroxymethy...)
Affinity DataKi:  505nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(GUINEA PIG)
Gilead Sciences

US Patent
LigandPNGBDBM377139(1-{9-[(4S,2R,3R,5R)-3,4-dihydroxy-5-(hydroxymethyl...)
Affinity DataKi: >1.00E+3nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(GUINEA PIG)
Gilead Sciences

US Patent
LigandPNGBDBM377137((4S,2R,3R,5R)-2-{6-Amino2-[4-(4-methylphenyl)pyraz...)
Affinity DataKi:  5.50E+3nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(GUINEA PIG)
Gilead Sciences

US Patent
LigandPNGBDBM377136((4S,2R,3R,5R)-2-{6-Amino-2-[4-(4-metboxyphenyl)pyr...)
Affinity DataKi:  5.50E+3nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(GUINEA PIG)
Gilead Sciences

US Patent
LigandPNGBDBM377135((4S,2R,3R,5R)-2-{6-Amino-2-[4-(4-chlorophenyl)pyra...)
Affinity DataKi:  5.50E+3nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(GUINEA PIG)
Gilead Sciences

US Patent
LigandPNGBDBM50152084(1-[6-Amino-9-(3,4-dihydroxy-5-hydroxymethyl-tetrah...)
Affinity DataKi:  5.50E+3nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
In DepthDetails US Patent