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Found 1 Enz. Inhib. hit(s) for PDB: 2AFZ
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

LigandPNGBDBM7942(1-Subsituted 1H-imidazole, 8 | 1-Vinylimidazole | ...)
Affinity DataKi:  4.90E+4nM ΔG°:  -25.0kJ/molepH: 8.0 T: 2°CAssay Description:QC activity was evaluated fluorometrically using Gln-AMC as substrate, and pyroglutamyl peptidase as the auxiliary enzyme. After conversion of Gln-AM...More data for this Ligand-Target Pair