Found 3 Enz. Inhib. hit(s) for PDB: 2CN8 TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 183nMAssay Description:Inhibition of human Chk2 using STK1 as substrate after 10 mins by HTRF assayMore data for this Ligand-Target Pair
3D Structure (crystal)TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 183nMAssay Description:Inhibition of CHK2 (unknown origin) using polypeptide substrate after 40 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of Chk2Checked by AuthorMore data for this Ligand-Target Pair
