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Found 1 Enz. Inhib. hit(s) for PDB: 2PE0
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Berlex Biosciences

LigandPNGBDBM17023((3Z)-5-hydroxy-3-[1-(1H-pyrrol-2-yl)ethylidene]-2,...)
Affinity DataIC50:  80nMpH: 7.2 T: 2°CAssay Description:The coupled assay can detect inhibitors of AKT2 activation, as well as direct inhibitors of PDK1 or AKT2. Inactive AKT2 is activated in situ by incub...More data for this Ligand-Target Pair