BindingDB PrimarySearch

Found 2 Enz. Inhib. hit(s) for PDB: 2VTJ

Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Astex

BDBM24631(4-[(6-chloropyrazin-2-yl)amino]benzene-1-sulfonami...)

IC50: 1.90E+3nMpH: 7.2 T: 2°CAssay Description:CDK2/cyclin A activity was determined using a radiometric assay to measure the incorporation of gamma-phosphate from [gamma-33P]-ATP into histone H1....More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar

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PDB

3D Structure (crystal)

Cyclin-dependent kinase 2(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL

BDBM24631(4-[(6-chloropyrazin-2-yl)amino]benzene-1-sulfonami...)

IC50: 9.10E+3nMAssay Description:Inhibition of CDK2More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Purchase CHEMBL DrugBank MMDB PC cid PC sid PDB

Details Article PubMed MMDB
PDB

3D Structure (crystal)