Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) for PDB: 2WMU
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
The Institute Of Cancer Research

LigandPNGBDBM33210(4-(7H-purin-6-yl)morpholine | purine, 9)
Affinity DataIC50:  4.20E+4nMpH: 7.5 T: 2°CAssay Description:CHK kinase function was measured in a DELFIA assay in order to monitor phosphorylation of a CDC25C peptide using a specific phospho antibody. The enz...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
The Institute Of Cancer Research

LigandPNGBDBM33210(4-(7H-purin-6-yl)morpholine | purine, 9)
Affinity DatapH: 7.5 T: 2°CAssay Description:AlphaScreen (PerkinElmer Life Sciences, Inc) was performed in opaque 384-well polypropylene plates. The assay relies on hydrogel coated Donor and Acc...More data for this Ligand-Target Pair