Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) for PDB: 3IDP
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Takeda California Inc

Curated by ChEMBL
LigandPNGBDBM35327(pyridylpurine aminoisoquinoline, 1)
Affinity DataKi:  1nMAssay Description:Inhibition of B-RafMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf [V600E](Homo sapiens (Human))
Amgen

LigandPNGBDBM35327(pyridylpurine aminoisoquinoline, 1)
Affinity DataIC50:  1.60nM EC50:  1.80nMpH: 7.0 T: 2°CAssay Description:The in vitro kinase activities of wild type or mutants were determined by measuring phosphorylation of biotinylated-MEK protein using Perkin-Elmer s ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Takeda California Inc

Curated by ChEMBL
LigandPNGBDBM35327(pyridylpurine aminoisoquinoline, 1)
Affinity DataIC50:  2nMAssay Description:Inhibition of b-Raf in human A375 cells assessed phosphorylation of ERKMore data for this Ligand-Target Pair