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Report error Found 3 Enz. Inhib. hit(s) for PDB: 3KDU
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50314814(2-((3-((2-(4-chlorophenyl)-5-methyloxazol-4-yl)met...)
Affinity DataIC50:  347nMAssay Description:Binding affinity to human His-tagged PPARalpha LBD (E196-Y468) expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50314814(2-((3-((2-(4-chlorophenyl)-5-methyloxazol-4-yl)met...)
Affinity DataEC50:  8.80nMAssay Description:Agonist activity at human PPARalpha LBD (167-468) expressed in HEK293 cells coexpressing GAL4-DBD by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50314814(2-((3-((2-(4-chlorophenyl)-5-methyloxazol-4-yl)met...)
Affinity DataEC50:  8nMAssay Description:Agonist activity against human Gal4-fussed PPARalpha in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)