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Found 3 Enz. Inhib. hit(s) for PDB: 3RM4
TargetAcidic mammalian chitinase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50378795(CHEMBL1215473)
Affinity DataIC50:  210nMAssay Description:Inhibition of acidic mammalian chitinase after 60 minsMore data for this Ligand-Target Pair
TargetAcidic mammalian chitinase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50378795(CHEMBL1215473)
Affinity DataIC50:  5.45E+3nMAssay Description:Inhibition of human recombinant full length C-terminal His-tagged acidic mammalian chitinase expressed in CHO-K1 cells using 4-methylumbelliferyl-bet...More data for this Ligand-Target Pair
TargetAcidic mammalian chitinase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50378795(CHEMBL1215473)
Affinity DataKd:  1.69E+3nMAssay Description:Binding affinity to biotinylated-acidic mammalian chitinaseMore data for this Ligand-Target Pair