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Report error Found 2 Enz. Inhib. hit(s) for PDB: 3V7R
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
Monash University

US Patent
LigandPNGBDBM161470(US9108978, 4.01)
Affinity DataKi:  660nM ΔG°:  -36.7kJ/mole IC50:  4.00E+3nMpH: 8.0 T: 37°CAssay Description:Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails US Patent
PDB3D3D Structure (crystal)

TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM161470(US9108978, 4.01)
Affinity DataKi:  660nMAssay Description:Inhibition of Staphylococcus aureus biotin protein ligase by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)