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Report error Found 3 Enz. Inhib. hit(s) for PDB: 4CI4
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti

Curated by ChEMBL
LigandPNGBDBM50401993(CHEMBL2204696)
Affinity DataEC50:  600nMAssay Description:Transactivation of human GAL4-fused PPARalpha ligand binding domain transfected in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti

Curated by ChEMBL
LigandPNGBDBM50401993(CHEMBL2204696)
Affinity DataEC50:  1.09E+3nMAssay Description:Agonist activity at Gal4-fused human PPARalpha LBD transfected in HEK293T cells assessed as transcriptional activation incubated for 14 to 16 hrs by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti

Curated by ChEMBL
LigandPNGBDBM50401993(CHEMBL2204696)
Affinity DataEC50:  2.10E+3nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)