Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) for PDB: 4DBS
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50382163(CHEMBL2023820)
Affinity DataIC50:  80nMAssay Description:Inhibition of recombinant AKR1C3 assessed as enzyme catalyzed oxidation of S-tetralol by fluorimetric assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C2(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50382163(CHEMBL2023820)
Affinity DataIC50:  8.17E+3nMAssay Description:Inhibition of recombinant AKR1C2 assessed as enzyme catalyzed oxidation of S-tetralol by fluorimetric assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C1(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50382163(CHEMBL2023820)
Affinity DataIC50:  1.11E+4nMAssay Description:Inhibition of recombinant AKR1C1 assessed as enzyme catalyzed oxidation of S-tetralol by fluorimetric assayMore data for this Ligand-Target Pair