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Found 3 Enz. Inhib. hit(s) for PDB: 4DMX
TargetCathepsin K(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50390404(CHEMBL2070936)
Affinity DataIC50:  15nMAssay Description:Inhibition of human recombinant cathepsin-k using Z-Phe-Arg-AMC as substrate preincubated for 15 mins measured after 1 hr by QFRET assayMore data for this Ligand-Target Pair
TargetCathepsin K(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50390404(CHEMBL2070936)
Affinity DataIC50:  15nMAssay Description:Inhibition of cathepsin-kMore data for this Ligand-Target Pair
TargetCathepsin K(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50390404(CHEMBL2070936)
Affinity DataIC50:  15.8nMAssay Description:Inhibition of human recombinant cathepsin K using Z-Phe-Arg-AMC as substrate preincubated for 30 mins measured after 1 hr by quenched fluorescent res...More data for this Ligand-Target Pair