BindingDB PrimarySearch_ki

Found 2 Enz. Inhib. hit(s) for PDB: 4LY9

Glucokinase regulatory protein(Homo sapiens (Human))
Amgen

Curated by ChEMBL

PNG

BDBM50447292(CHEMBL3113979)

IC50: 21nMAssay Description:Inhibition of biotin-tagged human GKRP-fluorescein-tagged human GK interaction preincubated for 20 mins followed by fluorescein-tagged human GK addit...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Details Article PubMed PDB

3D Structure (crystal)

Glucokinase regulatory protein(Rattus norvegicus)
Amgen

Curated by ChEMBL

PNG

BDBM50447292(CHEMBL3113979)

EC50: 82nMAssay Description:Inhibition of GKRP-GK interaction in rat primary hepatocytes assessed as translocation of GK from nucleus to cytoplasm preincubated for 20 mins follo...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

Purchase CHEMBL PC cid PC sid PDB Similars

Details Article PubMed PDB

3D Structure (crystal)