Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Bromodomain-containing protein 9 (105/105 = 100%)† (Homo sapiens (Human)) | BDBM50147621![]() (CHEMBL3769979) | PDB KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline R&D Curated by ChEMBL | Assay Description Inhibition of BRD9 in human HUT78 cells incubated for 45 mins by chemoproteomic competition binding assay | J Med Chem 59: 1425-39 (2016) Article DOI: 10.1021/acs.jmedchem.5b00256 BindingDB Entry DOI: 10.7270/Q2MS3VMP | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) |