Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Calmodulin-domain protein kinase 1 (CDPK1) (481/484 > 99%)† (Toxoplasma gondii) | BDBM286285![]() (US9518026, Example 78) | PDB UniProtKB/TrEMBL GoogleScholar | PC cid PC sid PDB UniChem | PDB US Patent | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Washington Through its Center For Commercialization US Patent | Assay Description Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti... | US Patent US9518026 (2016) | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) |