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Found 3 Enz. Inhib. hit(s) for PDB: 5CFW
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

LigandPNGBDBM188516(BDOIA383)
Affinity DataIC50:  2.40E+3nMAssay Description:The assay used a Cy5 dye-labeled BRD inhibitor PFI-411FP. The synthesis of the probe and the procedure for the assay was reported recently (Hett et a...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

LigandPNGBDBM188516(BDOIA383)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

LigandPNGBDBM188516(BDOIA383)
Affinity DataKd:  780nMAssay Description:Experiments were performed using recombinant CBP and BRD4 bromodomainsusing the procedure reported recently (Hett et al., 2015).More data for this Ligand-Target Pair