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Found 6 Enz. Inhib. hit(s) for PDB: 5FHM
TargetGlutamate receptor 3(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159745(CHEMBL3786901)
Affinity DataKi:  1.53E+3nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA3 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159745(CHEMBL3786901)
Affinity DataKi:  2.75E+3nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA4 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159745(CHEMBL3786901)
Affinity DataKi:  8.15E+3nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA2 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159745(CHEMBL3786901)
Affinity DataEC50:  1.29E+5nMAssay Description:Agonist activity at recombinant rat GluA4 receptor flip isoform expressed in Xenopus laevis oocytes by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159745(CHEMBL3786901)
Affinity DataEC50:  4.32E+5nMAssay Description:Agonist activity at recombinant rat GluA2(Q) receptor flip isoform expressed in Xenopus laevis oocytes by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
TargetGlutamate receptor 3(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159745(CHEMBL3786901)
Affinity DataEC50:  4.97E+4nMAssay Description:Agonist activity at recombinant rat GluA3 receptor flip isoform expressed in Xenopus laevis oocytes by two-electrode voltage clamp assayMore data for this Ligand-Target Pair