Found 1 Enz. Inhib. hit(s) for PDB: 5HE0 TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
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US Patent
The Regents Of The University Of Michigan
US Patent
Affinity DataIC50: 150nMpH: 7.0Assay Description:GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e...More data for this Ligand-Target Pair
3D Structure (crystal)