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Report error Found 6 Enz. Inhib. hit(s) for PDB: 5T8J
TargetAndrogen receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50238127(CHEMBL4092535)
Affinity DataIC50:  0.290nMAssay Description:Inhibition of rat liver pyruvate kinase (PK-L) at 7.2 mMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetAndrogen receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50238127(CHEMBL4092535)
Affinity DataIC50:  1nMAssay Description:Inhibition of Androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetAndrogen receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50238127(CHEMBL4092535)
Affinity DataIC50:  1nMAssay Description:Inhibition of rat liver pyruvate kinase (PK-L) at 10.7 mMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetAndrogen receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50238127(CHEMBL4092535)
Affinity DataIC50:  1nMAssay Description:Displacement of [3H]mibolerone from human AR after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetAndrogen receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50238127(CHEMBL4092535)
Affinity DataEC50:  0.290nMAssay Description:Modulation of Androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetAndrogen receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50238127(CHEMBL4092535)
Affinity DataEC50:  0.290nMAssay Description:Agonist activity at human AR expressed in African green monkey COS7 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)