Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 1 Enz. Inhib. hit(s) for PDB: 5VQK
TargetNuclear receptor ROR-gamma(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50549872(CHEMBL4792689)
Affinity DataIC50:  1.60E+3nMAssay Description:Antagonist activity at GAL4 DBD-fused human RORgamma LBD expressed in pGL4.3 luc2P/GAL4UAS/hygro and pBIND transfected HEK293 cells assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB