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Compile Data Set for Download or QSAR
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Found
1
Enz. Inhib. hit(s) for PDB:
5VQK
Target
Nuclear receptor ROR-gamma
(Human)
Boehringer Ingelheim Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50549872
(CHEMBL4792689)
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Affinity Data
IC50: 1.60E+3nM
Assay Description:
Antagonist activity at GAL4 DBD-fused human RORgamma LBD expressed in pGL4.3 luc2P/GAL4UAS/hygro and pBIND transfected HEK293 cells assessed as inhib...
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Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
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Ligand Info
PC cid
PC sid
PDB
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Details
Article
PubMed
PDB
3D Structure (crystal)
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