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Report error Found 2 Enz. Inhib. hit(s) for PDB: 5W0I
TargetCREB-binding protein(Human)
Genentech

Curated by ChEMBL
LigandPNGBDBM50269850(CHEMBL4061600)
Affinity DataIC50:  1.40nMAssay Description:Displacement of biotinylated histone H3K14 peptide ligand from human recombinant His-tagged CBP measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails
ArticlePubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein(Human)
Genentech

Curated by ChEMBL
LigandPNGBDBM50269850(CHEMBL4061600)
Affinity DataIC50:  37nMAssay Description:Inhibition of Halo-tagged histone H3.3 binding to NanoLuc luciferase conjugated human CBP expressed in HEK293 cells after overnight incubation by BRE...More data for this Ligand-Target Pair
In DepthDetails
ArticlePubMedPDB3D3D Structure (crystal)