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Report error Found 2 Enz. Inhib. hit(s) for PDB: 6E23
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50520121(CHEMBL4441671 | US10844044, Example 1)
Affinity DataKi:  0.0440nMAssay Description:Competitive inhibition of human N-terminal His6-SUMO tagged WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold(DE3) cells using 10-mer...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50520121(CHEMBL4441671 | US10844044, Example 1)
Affinity DataKi: <0.100nMAssay Description:A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo...More data for this Ligand-Target Pair
In DepthDetails US Patent
PDB3D3D Structure (crystal)