TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Membrane Research Group of The Hungarian Academy of Sciences
Curated by ChEMBL
Membrane Research Group of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:TP_TRANSPORTER: inhibition of ATPase activity in BCRP-expressing Sf9 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Membrane Research Group of The Hungarian Academy of Sciences
Curated by ChEMBL
Membrane Research Group of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:TP_TRANSPORTER: efflux of Hoechst33342 in BCRP-expressing Sf9 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Membrane Research Group of The Hungarian Academy of Sciences
Curated by ChEMBL
Membrane Research Group of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 3.38E+3nMAssay Description:Inhibition of BCRP expressed in MDCK cells by pheophorbide A assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Membrane Research Group of The Hungarian Academy of Sciences
Curated by ChEMBL
Membrane Research Group of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 3.71E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in human MCF7/MX cells mediated mitoxantrone efflux assessed as intracellular mitoxantrone level and m...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Membrane Research Group of The Hungarian Academy of Sciences
Curated by ChEMBL
Membrane Research Group of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.07E+3nMAssay Description:Inhibition of BCRP expressed in MCF7 MX cells by Hoechst 33342 stainingMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Membrane Research Group of The Hungarian Academy of Sciences
Curated by ChEMBL
Membrane Research Group of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of ABCG2 in human mitoxantrone-resistant MCF7 cells by Hoechst 33342 assayMore data for this Ligand-Target Pair