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Report error Found 2 Enz. Inhib. hit(s) for PDB: 7JXY
TargetTau-tubulin kinase 1(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50609146(CHEMBL5273263)
Affinity DataIC50:  18nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMedPDB3D3D Structure (crystal)

TargetTau-tubulin kinase 1(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50609146(CHEMBL5273263)
Affinity DataIC50:  259nMAssay Description:Inhibition of TTBK1 in human HEK293T cells incubated for 1 hrs by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMedPDB3D3D Structure (crystal)