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Report error Found 3 Enz. Inhib. hit(s) for PDB: 7WLN
TargetBromodomain-containing protein 2(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50604624(CHEMBL5206088)
Affinity DataIC50:  5.10nMAssay Description:Inhibition of C-terminal His6-tagged BRD2 BD2 (unknown origin) using H-YSGRGK(Ac)GGK(Ac)GLGK(Ac)-GGAK(Ac)RHRK-Biotin-OH as substrate incubated for 1 ...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50604624(CHEMBL5206088)
Affinity DataKd:  24nMAssay Description:Binding affinity to His6-fused BRD2 BD2 (unknown origin) assessed as dissociation constant in PBS incubated for 1 hrs by biolayer interferometry anal...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50604624(CHEMBL5206088)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to His6-fused BRD2 BD1 (unknown origin) assessed as dissociation constant in PBS incubated for 1 hrs by biolayer interferometry anal...More data for this Ligand-Target Pair