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Report error Found 2 Enz. Inhib. hit(s) for PDB: 7XNG
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50311438(CHEMBL4169942)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of biotinylated-H4KAc4 binding to human His6-tagged CBP (R1081 to G1197 residues) expressed in Escherichia coli BL21(DE3) after 2.5 hrs by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetHistone acetyltransferase p300(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50311438(CHEMBL4169942)
Affinity DataIC50:  2.51E+3nMAssay Description:Inhibition of biotinylated-H4KAc4 binding to human His6-tagged EP300 (A1040 to G1161 residues) expressed in Escherichia coli BL21(DE3) after 2.5 hrs ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)