TargetPeroxisome proliferator-activated receptor gamma(Human)
Institute of Mit and Harvard
Curated by ChEMBL
Institute of Mit and Harvard
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation in...More data for this Ligand-Target Pair
3D Structure (crystal)TargetPeroxisome proliferator-activated receptor gamma(Human)
Institute of Mit and Harvard
Curated by ChEMBL
Institute of Mit and Harvard
Curated by ChEMBL
Affinity DataEC50: 3.40nMAssay Description:Inverse agonist activity at GST tagged human PPARgamma LBD (231 to 505 residues) expressed in Escherichia coli BL21(DE3) assessed as recruitment of f...More data for this Ligand-Target Pair
