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Report error Found 3 Enz. Inhib. hit(s) for PDB: 8P5L
TargetSerine/threonine-protein kinase ULK1(Human)
Sichuan Universitt China Hospital

Curated by ChEMBL
LigandPNGBDBM50111572(CHEMBL3605057)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of GST-tagged ULK1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ULK1(Human)
Sichuan Universitt China Hospital

Curated by ChEMBL
LigandPNGBDBM50111572(CHEMBL3605057)
Affinity DataIC50:  45nMAssay Description:Inhibition of wild type GST-tagged ULK1 (unknown origin) after 5 mins in presence of gamma-[32]P-ATP by immunoblot analysisMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ULK1(Human)
Sichuan Universitt China Hospital

Curated by ChEMBL
LigandPNGBDBM50111572(CHEMBL3605057)
Affinity DataIC50:  170nMAssay Description:Inhibition of SUMO-tagged ULK1 (unknown origin) kinase domain expressed in KRX cells using [32P]-gamma-ATP and myelin basic protein substrate incubat...More data for this Ligand-Target Pair