Compile Data Set for Download or QSAR
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Found 10 Enz. Inhib. hit(s) with all data for entry = 50008498
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073876((1S,4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-met...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073875((1S,4S,5aS,9aS)-1,7,7-Tributyl-4-hydroxymethyl-5a-...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073873((1S,4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-1,5a-d...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073874((4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073874((4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073878((4R,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073872((4S,5aS,5bS,7aS,10aS,10bS,12aS)-4-Hydroxymethyl-5a...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073871((4R,5aS,5bS,7aS,10aS,10bS,12aS)-4-Hydroxymethyl-5a...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073877((4S,5aS,5bS,7aR,8R,10aS,10bR,12aS)-8-(1,5-Dimethyl...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073870((4R,5aS,5bS,7aR,8R,10aS,10bR,12aS)-8-(1,5-Dimethyl...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed