Compile Data Set for Download or QSAR
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Found 17 Enz. Inhib. hit(s) with all data for entry = 50008844
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077790((2S,3R,6S)-10-Benzenesulfonyl-4-oxo-3-(3-phenyl-pr...)
Affinity DataKi:  2nMAssay Description:Inhibition of Matrix metalloproteinase-9(MMP-9)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077789((2S,3R,6S)-4-Oxo-3-(3-phenyl-propyl)-1-oxa-5,10-di...)
Affinity DataKi:  4nMAssay Description:Inhibition of Matrix metalloproteinase-8(MMP-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077793((2S,3R,6S)-10-Acetyl-4-oxo-3-(3-phenyl-propyl)-1-o...)
Affinity DataKi:  6nMAssay Description:Inhibition of Matrix metalloproteinase-9(MMP-9)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077792((2S,3R,6S)-10-Acetyl-12-methyl-4-oxo-3-(3-phenyl-p...)
Affinity DataKi:  7nMAssay Description:Inhibition of Matrix metalloproteinase-8(MMP-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077791((2S,3R,6S)-2-Hydroxycarbamoyl-6-methylcarbamoyl-4-...)
Affinity DataKi:  13nMAssay Description:Inhibition of Matrix metalloproteinase-8(MMP-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077792((2S,3R,6S)-10-Acetyl-12-methyl-4-oxo-3-(3-phenyl-p...)
Affinity DataKi:  13nMAssay Description:Inhibition of Matrix metalloproteinase-9(MMP-9)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077791((2S,3R,6S)-2-Hydroxycarbamoyl-6-methylcarbamoyl-4-...)
Affinity DataKi:  19nMAssay Description:Inhibition of Matrix metalloproteinase-9(MMP-9)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077789((2S,3R,6S)-4-Oxo-3-(3-phenyl-propyl)-1-oxa-5,10-di...)
Affinity DataKi:  21nMAssay Description:Inhibition of Matrix metalloproteinase-9(MMP-9)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077793((2S,3R,6S)-10-Acetyl-4-oxo-3-(3-phenyl-propyl)-1-o...)
Affinity DataKi:  38nMAssay Description:Inhibition of Matrix metalloproteinase-3(MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077790((2S,3R,6S)-10-Benzenesulfonyl-4-oxo-3-(3-phenyl-pr...)
Affinity DataKi:  110nMAssay Description:Inhibition of Matrix metalloproteinase-1(MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077793((2S,3R,6S)-10-Acetyl-4-oxo-3-(3-phenyl-propyl)-1-o...)
Affinity DataKi:  248nMAssay Description:Inhibition of Matrix metalloproteinase-1(MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077789((2S,3R,6S)-4-Oxo-3-(3-phenyl-propyl)-1-oxa-5,10-di...)
Affinity DataKi:  265nMAssay Description:Inhibition of Matrix metalloproteinase-3(MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077792((2S,3R,6S)-10-Acetyl-12-methyl-4-oxo-3-(3-phenyl-p...)
Affinity DataKi:  267nMAssay Description:Inhibition of Matrix metalloproteinase-3(MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077791((2S,3R,6S)-2-Hydroxycarbamoyl-6-methylcarbamoyl-4-...)
Affinity DataKi:  373nMAssay Description:Inhibition of Matrix metalloproteinase-3(MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077792((2S,3R,6S)-10-Acetyl-12-methyl-4-oxo-3-(3-phenyl-p...)
Affinity DataKi:  440nMAssay Description:Inhibition of Matrix metalloproteinase-1(MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077789((2S,3R,6S)-4-Oxo-3-(3-phenyl-propyl)-1-oxa-5,10-di...)
Affinity DataKi:  496nMAssay Description:Inhibition of Matrix metalloproteinase-1(MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50077791((2S,3R,6S)-2-Hydroxycarbamoyl-6-methylcarbamoyl-4-...)
Affinity DataKi:  1.07E+3nMAssay Description:Inhibition of Matrix metalloproteinase-1(MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed