Affinity DataKi: 9.40nMAssay Description:In vitro binding affinity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:In vitro binding affinity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:In vitro binding affinity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:In vitro binding affinity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:In vitro binding affinity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:In vitro binding affinity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:In vitro binding affinity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 139nMAssay Description:In vitro binding affinity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataEC50: 0.25nMAssay Description:In vitro intrinsic activity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:In vitro intrinsic activity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataEC50: 0.220nMAssay Description:In vitro intrinsic activity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataEC50: 128nMAssay Description:In vitro binding affinity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataEC50: 2.80nMAssay Description:In vitro binding affinity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:In vitro binding affinity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataEC50: 0.550nMAssay Description:In vitro intrinsic activity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair