Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50036766
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50082524(2,6-Bis(3-pyrrolidinopropionamido)anthracene-9,10-...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080847(3,6-Bis(3-piperidinopropionamido)acridine | 3-Pipe...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080840(3,6-Bis[3-(azepan-1-yl)propionamido]acridine | 3,6...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50082532(2,6-Bis(3-piperidinopropionamido)anthracene-9,10-d...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080849(3,6-Bis(3-pyrrolidinopropionamido)acridine | 3-PYR...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50082530(2,6-Bis[3-(hexamethyleneimino)propionamido]anthrac...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080852(3,6-Bis[3-(heptamethyleneimino)piperizinopropionam...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50082526(2,6-Bis[3-(1,3,3-trimethyl-6-azabicyclo[3.2.1]octa...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080846(3,6-Bis[3-(1,3,3-trimethyl-6-azabicyclo[3.2.1]octa...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50082528(2,6-Bis[3-(heptamethyleneimino)propionamido]anthra...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed